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Found 175 with Last Name = 'mitani' and Initial = 'h'
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50348228(CHEMBL1800807)
Affinity DataIC50:  18nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50312718(CHEMBL479527 | torcetrapib)
Affinity DataIC50:  18nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250371(CHEMBL4064793)
Affinity DataIC50:  60nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250366(CHEMBL4075773)
Affinity DataIC50:  62nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250363(CHEMBL4070653)
Affinity DataIC50:  71nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218471(4-[7,7,10,10-tetramethyl-5-propyl-2-(3-trifluorome...)
Affinity DataIC50:  76nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218455(4-[5-ethyl-7,7,10,10-tetramethyl-2-(3-trifluoromet...)
Affinity DataIC50:  95nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50381415(EVACETRAPIB | LY2484595)
Affinity DataIC50:  110nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218481(4-[2-(4-fluoro-benzenesulfonylamino)-7,7,10,10-tet...)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218438(4-[5,7,7,10,10-pentamethyl-2-(4-trifluoromethoxy-b...)
Affinity DataIC50:  130nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218461(4-[2-(butane-1-sulfonylamino)-7,7,10,10-tetramethy...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250365(CHEMBL4103344)
Affinity DataIC50:  150nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218455(4-[5-ethyl-7,7,10,10-tetramethyl-2-(3-trifluoromet...)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250355(CHEMBL4081265)
Affinity DataIC50:  160nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250355(CHEMBL4081265)
Affinity DataIC50:  160nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250364(CHEMBL4063323)
Affinity DataIC50:  164nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250364(CHEMBL4063323)
Affinity DataIC50:  164nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218429(4-[2-(4-methoxy-benzenesulfonyl)-5,7,7,10,10-penta...)
Affinity DataIC50:  170nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218471(4-[7,7,10,10-tetramethyl-5-propyl-2-(3-trifluorome...)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218468(4-[2-(4-fluoro-benzenesulfonylamino)-5,7,7,10,10-p...)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218448(4-(2-butylsulfamoyl-5,7,7,10,10-pentamethyl-7,8,9,...)
Affinity DataIC50:  190nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250370(CHEMBL4083767)
Affinity DataIC50:  200nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218458(4-[2-(butane-1-sulfonylamino)-5-ethyl-7,7,10,10-te...)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218492(4-[5-ethyl-2-(4-fluoro-benzenesulfonylamino)-7,7,1...)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250357(CHEMBL4089133)
Affinity DataIC50:  240nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218438(4-[5,7,7,10,10-pentamethyl-2-(4-trifluoromethoxy-b...)
Affinity DataIC50:  240nMAssay Description:Inhibition of LG100268-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218495(4-[5,7,7,10,10-pentamethyl-2-(propane-1-sulfonylam...)
Affinity DataIC50:  250nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218433(4-(2-cyano-5-ethyl-7,7,10,10-tetramethyl-7,8,9,10-...)
Affinity DataIC50:  320nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218458(4-[2-(butane-1-sulfonylamino)-5-ethyl-7,7,10,10-te...)
Affinity DataIC50:  320nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218454(4-[5-ethyl-7,7,10,10-tetramethyl-2-(propane-1-sulf...)
Affinity DataIC50:  340nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218429(4-[2-(4-methoxy-benzenesulfonyl)-5,7,7,10,10-penta...)
Affinity DataIC50:  360nMAssay Description:Inhibition of LG100268-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218469(4-[2-(butane-1-sulfonylamino)-5,7,7,10,10-pentamet...)
Affinity DataIC50:  370nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218434(4-[5,7,7,10,10-pentamethyl-2-(4-trifluoromethoxy-p...)
Affinity DataIC50:  390nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218496(4-[5,7,7,10,10-pentamethyl-2-((E)-2-phenyl-ethenes...)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218448(4-(2-butylsulfamoyl-5,7,7,10,10-pentamethyl-7,8,9,...)
Affinity DataIC50:  410nMAssay Description:Inhibition of LG100268-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218446(4-[2-(4-chloro-phenylmethanesulfonyl)-5,7,7,10,10-...)
Affinity DataIC50:  420nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218492(4-[5-ethyl-2-(4-fluoro-benzenesulfonylamino)-7,7,1...)
Affinity DataIC50:  420nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218436(4-(2-cyano-5,7,7,10,10-pentamethyl-7,8,9,10-tetrah...)
Affinity DataIC50:  430nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218499(4-[5,7,7,10,10-pentamethyl-2-(toluene-4-sulfonylam...)
Affinity DataIC50:  430nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218428(4-[5,7,7,10,10-pentamethyl-2-(morpholine-4-sulfony...)
Affinity DataIC50:  450nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218444(4-[5,7,7,10,10-pentamethyl-2-(pyrrolidine-1-sulfon...)
Affinity DataIC50:  450nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218453(4-[5,7,7,10,10-pentamethyl-2-(propane-1-sulfonyl)-...)
Affinity DataIC50:  450nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218427(4-[5,7,7,10,10-pentamethyl-2-(4-trifluoromethoxy-p...)
Affinity DataIC50:  460nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218490(4-[2-(4-methoxy-benzenesulfonylamino)-5,7,7,10,10-...)
Affinity DataIC50:  470nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218433(4-(2-cyano-5-ethyl-7,7,10,10-tetramethyl-7,8,9,10-...)
Affinity DataIC50:  480nMAssay Description:Inhibition of LG100268-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218456(4-[5,7,7,10,10-pentamethyl-2-(3-trifluoromethyl-be...)
Affinity DataIC50:  480nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218424(4-(2-cyano-5-ethyl-7,7,10,10-tetramethyl-7,8,9,10-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218466(4-(2-benzenesulfonylamino-5,7,7,10,10-pentamethyl-...)
Affinity DataIC50:  510nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250359(CHEMBL4074770)
Affinity DataIC50:  510nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218432(4-(2-cyano-5,7,7,10,10-pentamethyl-7,8,9,10-tetrah...)
Affinity DataIC50:  520nMAssay Description:Inhibition of 9-cis-retinoic acid-induced RXRalpha transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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