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Found 176 with Last Name = 'mitscher' and Initial = 'la'
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kansas University

Curated by ChEMBL
LigandPNGBDBM50366826(DR-3355 | Floxacin | Iquix | LEVOFLOXACIN | Levaqu...)
Affinity DataKi:  2.49E+3nMAssay Description:Binding affinity against sigma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kansas University

Curated by ChEMBL
LigandPNGBDBM50045000((NFLX)1-Ethyl-6-fluoro-4-oxo-7-piperazin-1-yl-1,4-...)
Affinity DataKi:  3.13E+3nMAssay Description:Binding affinity against sigma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kansas University

Curated by ChEMBL
LigandPNGBDBM50045004(9-fluoro-3-methyl-10-(4-methylpiperazin-1-yl)-7-ox...)
Affinity DataKi:  4.42E+3nMAssay Description:Binding affinity for dopamine receptor D2 was evaluated by the ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kansas University

Curated by ChEMBL
LigandPNGBDBM50226409(DEXTROFLOXACINE)
Affinity DataKi:  7.47E+4nMAssay Description:Binding affinity against sigma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kansas University

Curated by ChEMBL
LigandPNGBDBM50366826(DR-3355 | Floxacin | Iquix | LEVOFLOXACIN | Levaqu...)
Affinity DataKi:  9.96E+4nMAssay Description:Binding affinity for dopamine receptor D2 was evaluated by the ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kansas University

Curated by ChEMBL
LigandPNGBDBM50045000((NFLX)1-Ethyl-6-fluoro-4-oxo-7-piperazin-1-yl-1,4-...)
Affinity DataKi:  2.25E+5nMAssay Description:Binding affinity for dopamine receptor D2 was evaluated by the ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kansas University

Curated by ChEMBL
LigandPNGBDBM50045004(9-fluoro-3-methyl-10-(4-methylpiperazin-1-yl)-7-ox...)
Affinity DataKi:  2.32E+5nMAssay Description:Binding affinity against sigma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kansas University

Curated by ChEMBL
LigandPNGBDBM50226409(DEXTROFLOXACINE)
Affinity DataKi:  2.90E+5nMAssay Description:Binding affinity against sigma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383959(CHEMBL2031999)
Affinity DataIC50:  10nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481476(CHEMBL599404)
Affinity DataIC50:  40nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481462(CHEMBL597782)
Affinity DataIC50:  40nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383948(CHEMBL2031983)
Affinity DataIC50:  40nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50481859(CHEMBL1088309)
Affinity DataIC50:  50nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481477(CHEMBL599402)
Affinity DataIC50:  50nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50481859(CHEMBL1088309)
Affinity DataIC50:  50nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481448(CHEMBL605965)
Affinity DataIC50:  50nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481480(CHEMBL599829)
Affinity DataIC50:  60nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481472(CHEMBL597585)
Affinity DataIC50:  70nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50017702(1-(bis(4-fluorophenyl)methyl)-4-cinnamylpiperazine...)
Affinity DataIC50:  80nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50095765(1-(2,3,4-trimethoxybenzyl)-4-(bis(4-fluorophenyl)m...)
Affinity DataIC50:  90nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50481862(CHEMBL1087275)
Affinity DataIC50:  90nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50481860(CHEMBL1087660)
Affinity DataIC50:  90nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481475(CHEMBL598592)
Affinity DataIC50:  90nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383936(CHEMBL2031965)
Affinity DataIC50:  100nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481493(CHEMBL597783)
Affinity DataIC50:  100nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383962(CHEMBL2031961)
Affinity DataIC50:  100nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383939(CHEMBL2031969)
Affinity DataIC50:  100nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383945(CHEMBL2031980)
Affinity DataIC50:  100nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383946(CHEMBL2031981)
Affinity DataIC50:  100nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383947(CHEMBL2031982)
Affinity DataIC50:  100nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383958(CHEMBL2031998)
Affinity DataIC50:  100nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481486(CHEMBL597788)
Affinity DataIC50:  110nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481470(CHEMBL596946)
Affinity DataIC50:  110nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50461289(MK-6721 | NMED-160 | NP-118809 | Z-160 | Z160)
Affinity DataIC50:  110nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50481858(CHEMBL1086621)
Affinity DataIC50:  110nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50461289(MK-6721 | NMED-160 | NP-118809 | Z-160 | Z160)
Affinity DataIC50:  110nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50481447(CHEMBL598598)
Affinity DataIC50:  110nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383960(CHEMBL2032000)
Affinity DataIC50:  110nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zalicus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50383938(CHEMBL2031967)
Affinity DataIC50:  130nMAssay Description:Inhibition of human Erg expressed in HEK293 cells by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50481868(CHEMBL1088610)
Affinity DataIC50:  130nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481484(CHEMBL599403)
Affinity DataIC50:  140nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481451(CHEMBL599821)
Affinity DataIC50:  140nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50481864(CHEMBL1087237)
Affinity DataIC50:  150nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481466(CHEMBL599217)
Affinity DataIC50:  150nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50481466(CHEMBL599217)
Affinity DataIC50:  150nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481482(CHEMBL598806)
Affinity DataIC50:  170nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-1(Homo sapiens)
Neuromed Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50481474(CHEMBL603465)
Affinity DataIC50:  180nMAssay Description:Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50481861(CHEMBL1087779)
Affinity DataIC50:  190nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50481863(CHEMBL1088464)
Affinity DataIC50:  190nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50481869(CHEMBL1088308)
Affinity DataIC50:  190nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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