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Found 160 with Last Name = 'miyadera' and Initial = 'k'
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376962(US10329300, Example 50 | US11696917, Example 50 | ...)
Affinity DataIC50:  2.90nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376962(US10329300, Example 50 | US11696917, Example 50 | ...)
Affinity DataIC50:  2.90nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376933(US10329300, Example 27 | US11696917, Example 27 | ...)
Affinity DataIC50:  3.90nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376933(US10329300, Example 27 | US11696917, Example 27 | ...)
Affinity DataIC50:  3.90nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376912(US10329300, Example 6 | US11696917, Example 6 | US...)
Affinity DataIC50:  4nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376912(US10329300, Example 6 | US11696917, Example 6 | US...)
Affinity DataIC50:  4nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376924(US10329300, Example 18 | US11696917, Example 18 | ...)
Affinity DataIC50:  4.40nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376924(US10329300, Example 18 | US11696917, Example 18 | ...)
Affinity DataIC50:  4.40nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376920(US10329300, Example 14 | US11696917, Example 14 | ...)
Affinity DataIC50:  4.60nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376920(US10329300, Example 14 | US11696917, Example 14 | ...)
Affinity DataIC50:  4.60nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376988(US10329300, Example 76 | US11696917, Example 76 | ...)
Affinity DataIC50:  5nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376988(US10329300, Example 76 | US11696917, Example 76 | ...)
Affinity DataIC50:  5nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376948(US10329300, Example 36 | US11696917, Example 36 | ...)
Affinity DataIC50:  5.40nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376948(US10329300, Example 36 | US11696917, Example 36 | ...)
Affinity DataIC50:  5.40nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376923(US10329300, Example 17 | US11696917, Example 17 | ...)
Affinity DataIC50:  5.90nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376923(US10329300, Example 17 | US11696917, Example 17 | ...)
Affinity DataIC50:  5.90nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376945((R)-4-(1-(1-acryloylpiperidin-3-yl)-4-amino-1H-pyr...)
Affinity DataIC50:  6nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376945((R)-4-(1-(1-acryloylpiperidin-3-yl)-4-amino-1H-pyr...)
Affinity DataIC50:  6nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376941(US10329300, Example 29 | US11696917, Example 29 | ...)
Affinity DataIC50:  6.5nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376941(US10329300, Example 29 | US11696917, Example 29 | ...)
Affinity DataIC50:  6.5nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376932(US10329300, Example 26 | US11696917, Example 26 | ...)
Affinity DataIC50:  7nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376932(US10329300, Example 26 | US11696917, Example 26 | ...)
Affinity DataIC50:  7nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376913(US10329300, Example 7 | US11696917, Example 7 | US...)
Affinity DataIC50:  7.10nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376909(US10329300, Example 3 | US9920060, 3)
Affinity DataIC50:  7.10nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376909(US10329300, Example 3 | US9920060, 3)
Affinity DataIC50:  7.10nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376913(US10329300, Example 7 | US11696917, Example 7 | US...)
Affinity DataIC50:  7.10nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376918(US10329300, Example 12 | US11696917, Example 12 | ...)
Affinity DataIC50:  7.5nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376917(US10329300, Example 11 | US11696917, Example 11 | ...)
Affinity DataIC50:  7.5nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376918(US10329300, Example 12 | US11696917, Example 12 | ...)
Affinity DataIC50:  7.5nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376917(US10329300, Example 11 | US11696917, Example 11 | ...)
Affinity DataIC50:  7.5nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376980((R)-4-(1-(1-acryloylpyrimidin-3-yl)-4-amino-1H-pyr...)
Affinity DataIC50:  7.70nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376980((R)-4-(1-(1-acryloylpyrimidin-3-yl)-4-amino-1H-pyr...)
Affinity DataIC50:  7.70nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376908(US10329300, Example 2 | US9920060, 2)
Affinity DataIC50:  8.30nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376908(US10329300, Example 2 | US9920060, 2)
Affinity DataIC50:  8.30nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376960(US10329300, Example 48 | US11696917, Example 48 | ...)
Affinity DataIC50:  8.5nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376960(US10329300, Example 48 | US11696917, Example 48 | ...)
Affinity DataIC50:  8.5nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376921(US10329300, Example 15 | US11696917, Example 15 | ...)
Affinity DataIC50:  8.60nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376921(US10329300, Example 15 | US11696917, Example 15 | ...)
Affinity DataIC50:  8.60nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376942(US10329300, Example 30 | US11696917, Example 30 | ...)
Affinity DataIC50:  8.70nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376942(US10329300, Example 30 | US11696917, Example 30 | ...)
Affinity DataIC50:  8.70nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376914(US10329300, Example 8 | US11696917, Example 8 | US...)
Affinity DataIC50:  9.20nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376981(US11696917, Example 69 | US9920060, 69)
Affinity DataIC50:  9.20nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376914(US10329300, Example 8 | US11696917, Example 8 | US...)
Affinity DataIC50:  9.20nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376944(US10329300, Example 32 | US11696917, Example 32 | ...)
Affinity DataIC50:  9.30nMAssay Description:For setting the conditions for the method for measuring the in vitro inhibitory activity of a compound against HER2-phosphorylating activity, Profile...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376944(US10329300, Example 32 | US11696917, Example 32 | ...)
Affinity DataIC50:  9.30nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376907(US10329300, Example 1 | US9920060, 1)
Affinity DataIC50:  10nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376915(US10329300, Example 9 | US11696917, Example 9 | US...)
Affinity DataIC50:  10nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376922(US10329300, Example 16 | US11696917, Example 16 | ...)
Affinity DataIC50:  10nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376925(US10329300, Example 19 | US11696917, Example 19 | ...)
Affinity DataIC50:  10nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM376950(US10329300, Example 38 | US11696917, Example 38 | ...)
Affinity DataIC50:  10nMAssay Description:For the inhibitory activity measurement of each compound, the compound of the present invention or staurosporine was first serially diluted with dime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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