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Found 130 with Last Name = 'miyagawa' and Initial = 'h'
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | CHEM...)
Affinity DataIC50:  1.29nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
TargetBeta-glucuronidase(Homo sapiens (Human))TBA
LigandPNGBDBM50405568(CHEMBL5273557)
Affinity DataIC50:  9.80nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50:  45.7nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414658(CHEMBL559048)
Affinity DataIC50:  58.9nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414645(CYASTERONE)
Affinity DataIC50:  61.7nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414646(INOKOSTERONE)
Affinity DataIC50:  91.2nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50226672(CHEMBL255034 | makisterone A)
Affinity DataIC50:  112nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414659(CHEMBL564892)
Affinity DataIC50:  324nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414652(CHEMBL559941)
Affinity DataIC50:  794nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488465(CHEMBL2286413)
Affinity DataIC50:  2.24E+3nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414651(ECDYSONE)
Affinity DataIC50:  2.57E+3nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405568(CHEMBL5273557)
Affinity DataIC50:  3.41E+3nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405566(CHEMBL5284745)
Affinity DataIC50:  4.04E+3nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405569(CHEMBL5276305)
Affinity DataIC50:  7.89E+3nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405570(CHEMBL5280906)
Affinity DataIC50:  8.03E+3nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488464(CHEMBL2286419)
Affinity DataIC50:  8.91E+3nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405558(CHEMBL3347523)
Affinity DataIC50:  9.19E+3nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414655(CHEMBL560796)
Affinity DataIC50:  9.55E+3nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405567(CHEMBL5280810)
Affinity DataIC50:  1.12E+4nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405559(CHEMBL5290753)
Affinity DataIC50:  1.20E+4nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488463(CHEMBL2285681)
Affinity DataIC50:  1.29E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488463(CHEMBL2285681)
Affinity DataIC50:  1.35E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414657(CHEMBL562711)
Affinity DataIC50:  1.45E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488437(CHEMBL2286416)
Affinity DataIC50:  1.48E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488465(CHEMBL2286413)
Affinity DataIC50:  1.51E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488447(CHEMBL2286412)
Affinity DataIC50:  1.62E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405560(CHEMBL5281456)
Affinity DataIC50:  1.92E+4nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405561(CHEMBL5273519)
Affinity DataIC50:  1.93E+4nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405565(CHEMBL5279462)
Affinity DataIC50:  1.97E+4nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405563(CHEMBL5283021)
Affinity DataIC50:  2.15E+4nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488448(CHEMBL2286411)
Affinity DataIC50:  2.40E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488438(CHEMBL2286414)
Affinity DataIC50:  2.40E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488438(CHEMBL2286414)
Affinity DataIC50: <2.51E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488477(CHEMBL2286417)
Affinity DataIC50:  2.69E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488448(CHEMBL2286411)
Affinity DataIC50:  2.82E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405562(CHEMBL5270267)
Affinity DataIC50:  3.05E+4nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414660(CHEMBL564474)
Affinity DataIC50:  3.89E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414647(CHEMBL560194)
Affinity DataIC50:  4.17E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414649(CHEMBL561275)
Affinity DataIC50:  4.17E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488462(CHEMBL2286415)
Affinity DataIC50:  4.79E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))TBA
LigandPNGBDBM50405564(CHEMBL4650593)
Affinity DataIC50:  5.01E+4nMAssay Description:In vitro concentration required to inhibit partially purified dihydropteroate synthase of Escherichia coli by 50%More data for this Ligand-Target Pair
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488462(CHEMBL2286415)
Affinity DataIC50:  5.50E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488447(CHEMBL2286412)
Affinity DataIC50:  6.76E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488477(CHEMBL2286417)
Affinity DataIC50:  7.41E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488437(CHEMBL2286416)
Affinity DataIC50:  7.94E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414653(CHEMBL558256)
Affinity DataIC50:  8.91E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414648(CHEMBL559545)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414654(CHEMBL560139)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414656(CHEMBL558652)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414650(CHEMBL550600)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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