Affinity DataIC50: 31nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 154nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 159nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 192nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 203nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 305nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 325nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 337nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 594nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 663nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: >2.40E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.21E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at human S1P3 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at human S1P4 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >8.10E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+4nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Antagonist activity at human S1P2 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at human S1P3 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair