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Found 197 with Last Name = 'mizuno' and Initial = 'y'
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208895(CHEMBL397081 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135494(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  56nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208889(sodium 4-[(4-butoxyphenyl)thio]-20-(1,12-dihydroxy...)
Affinity DataIC50:  80nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135493(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50:  82nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208901(CHEMBL239876 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  98nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208900(CHEMBL396365 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135496(CHEMBL130156 | [4-(5-Fluoro-3-methyl-benzo[b]thiop...)
Affinity DataIC50:  154nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135499(2-[4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfon...)
Affinity DataIC50:  159nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208884(CHEMBL241104 | sodium 20-(1-hydroxytridec-2-yn-1-y...)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208887(CHEMBL239659 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135509(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50:  192nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135495(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  203nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135502(3-Methanesulfonyl-4-(3-methyl-benzo[b]thiophene-2-...)
Affinity DataIC50:  305nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135497(4-(3,5-Dimethyl-benzo[b]thiophene-2-sulfonylamino)...)
Affinity DataIC50:  325nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135506(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50:  337nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208896(CHEMBL397080 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  340nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208897(CHEMBL239874 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  370nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208888(CHEMBL239867 | sodium 4-(4-ethoxyphenoxy)-20-(1-hy...)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208886(CHEMBL239653 | sodium 4-[(4-ethoxyphenyl)thio]-20-...)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208895(CHEMBL397081 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208894(CHEMBL277377 | sodium 4-[(4-hexyloxyphenyl)thio]-2...)
Affinity DataIC50:  520nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135501(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  594nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135505(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  663nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208882(CHEMBL240079 | sodium 20-(1-hydroxytridec-2-yn-1-y...)
Affinity DataIC50:  700nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135507(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  880nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135494(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135508(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135495(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135503(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135493(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135494(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135493(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135495(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208893(CHEMBL396847 | sodium 4-(4-ethoxyphenoxy)-20-(1-hy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135498(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208887(CHEMBL239659 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208883(CHEMBL429810 | sodium 2-(4-ethoxyphenoxy)-5-[3-(1-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135504(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  1.65E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208903(CHEMBL239873 | sodium 4-[(4-octyloxyphenyl)thio]-2...)
Affinity DataIC50: >2.40E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135500(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  4.21E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208899(CHEMBL239650 | sodium 4-(4-ethoxyphenoxy)-30-(1-hy...)
Affinity DataIC50:  4.60E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208895(CHEMBL397081 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at human S1P3 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208891(CHEMBL240078 | sodium 2-(4-ethoxyphenoxy)-5-[5-(1-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208895(CHEMBL397081 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  6.00E+3nMAssay Description:Antagonist activity at human S1P4 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208892(20-(1-aminotridec-2-yn-1-yl)-4-[(4-butoxyphenyl)th...)
Affinity DataIC50: >8.10E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208898(CHEMBL399392 | sodium 4-(2-ethoxyphenoxy)-20-(1-hy...)
Affinity DataIC50:  8.90E+3nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50121657(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50:  1.06E+4nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 2(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208895(CHEMBL397081 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  1.10E+4nMAssay Description:Antagonist activity at human S1P2 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208887(CHEMBL239659 | sodium 4-[(4-butoxyphenyl)thio]-20-...)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at human S1P3 receptor expressed in CHO cell membrane by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50208902(2-(4-ethoxyphenoxy)-5-(3-octadecyl-5-oxo-4,5-dihyd...)
Affinity DataIC50:  1.70E+4nMAssay Description:Antagonist activity at human S1P1 receptor expressed in CHO cell membrane by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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