TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 1.86nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 4.57nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 5.01nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 7.76nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 9.12nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 11.0nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 12.3nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 15.5nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 23.4nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 26.3nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 50.1nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Antagonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as inhibition of increase in intracellular calcium compound pr...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of C3 cleavage in human serum assessed as reduction in C5b-9 formation compound preincubated for 15 mins measured 1 hr post LPS stimulatio...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of C3 cleavage in human serum assessed as reduction in C3b formation compound preincubated for 15 mins measured 1 hr post LPS stimulation ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 8.91E+3nMAssay Description:Antagonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as inhibition of increase in intracellular calcium compound pr...More data for this Ligand-Target Pair
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.31E+4nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.78E+4nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 5.36E+4nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.32E+5nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+5nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration for human complement component C3 activationMore data for this Ligand-Target Pair