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Found 272 with Last Name = 'morimoto' and Initial = 'h'
TargetEndothelin-1 receptor(Homo sapiens (Human))
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105033(CHEMBL112531 | N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)...)
Affinity DataKi:  0.00420nMAssay Description:Ability to inhibit [125I]ET1 binding to human cloned endothelin A receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50369953(CHEMBL1627022)
Affinity DataKi:  0.0150nMAssay Description:Ability to inhibit [125I]ET1 binding to human cloned endothelin A receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088846(CHEMBL353678 | N-{4-[2-(4-Phenyl-piperazin-1-yl)-e...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088844(4-{4-[4-(4-Phenyl-piperazin-1-yl)-butyl]-phenyl}-t...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088839(CHEMBL169702 | N-{4-[4-(4-Phenyl-piperazin-1-yl)-b...)
Affinity DataKi:  4.60nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088844(4-{4-[4-(4-Phenyl-piperazin-1-yl)-butyl]-phenyl}-t...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088839(CHEMBL169702 | N-{4-[4-(4-Phenyl-piperazin-1-yl)-b...)
Affinity DataKi:  6nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088841(CHEMBL352617 | N-{4-[3-(4-Phenyl-piperazin-1-yl)-p...)
Affinity DataKi:  6.40nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088844(4-{4-[4-(4-Phenyl-piperazin-1-yl)-butyl]-phenyl}-t...)
Affinity DataKi:  7.90nMAssay Description:Inhibition of class C beta-lactamase derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088841(CHEMBL352617 | N-{4-[3-(4-Phenyl-piperazin-1-yl)-p...)
Affinity DataKi:  33nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088844(4-{4-[4-(4-Phenyl-piperazin-1-yl)-butyl]-phenyl}-t...)
Affinity DataKi:  37nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50369953(CHEMBL1627022)
Affinity DataKi:  41nMAssay Description:Ability to inhibit [125I]-ET-1 binding to human cloned ETB receptors expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088839(CHEMBL169702 | N-{4-[4-(4-Phenyl-piperazin-1-yl)-b...)
Affinity DataKi:  48nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088839(CHEMBL169702 | N-{4-[4-(4-Phenyl-piperazin-1-yl)-b...)
Affinity DataKi:  49nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088846(CHEMBL353678 | N-{4-[2-(4-Phenyl-piperazin-1-yl)-e...)
Affinity DataKi:  69nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105000(CHEMBL175616 | sodium salt of 4-tert-Butyl-N-[6-(2...)
Affinity DataKi:  81nMAssay Description:Ability to inhibit [125I]ET1 binding to human cloned endothelin A receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088846(CHEMBL353678 | N-{4-[2-(4-Phenyl-piperazin-1-yl)-e...)
Affinity DataKi:  130nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105033(CHEMBL112531 | N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)...)
Affinity DataKi:  130nMAssay Description:Ability to inhibit [125I]-ET-1 binding to human cloned ETB receptors expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088845(CHEMBL170307 | N-[4-(4-Phenyl-piperazin-1-ylmethyl...)
Affinity DataKi:  140nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105000(CHEMBL175616 | sodium salt of 4-tert-Butyl-N-[6-(2...)
Affinity DataKi:  140nMAssay Description:Ability to inhibit [125I]-ET-1 binding to human cloned ETB receptors expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088841(CHEMBL352617 | N-{4-[3-(4-Phenyl-piperazin-1-yl)-p...)
Affinity DataKi:  160nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088846(CHEMBL353678 | N-{4-[2-(4-Phenyl-piperazin-1-yl)-e...)
Affinity DataKi:  170nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088841(CHEMBL352617 | N-{4-[3-(4-Phenyl-piperazin-1-yl)-p...)
Affinity DataKi:  340nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088843(CHEMBL171115 | N-{4-[4-(4-Methoxy-phenyl)-piperazi...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088840(CHEMBL352576 | N-{4-[4-(2,4-Difluoro-phenyl)-piper...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088845(CHEMBL170307 | N-[4-(4-Phenyl-piperazin-1-ylmethyl...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro inhibition of human plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088842(CHEMBL171052 | N-{4-[4-(4-Fluoro-phenyl)-piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088843(CHEMBL171115 | N-{4-[4-(4-Methoxy-phenyl)-piperazi...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088843(CHEMBL171115 | N-{4-[4-(4-Methoxy-phenyl)-piperazi...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088842(CHEMBL171052 | N-{4-[4-(4-Fluoro-phenyl)-piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088847(CHEMBL171345 | N-{4-[4-(4-Chloro-phenyl)-piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of class C beta-lactamase derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088840(CHEMBL352576 | N-{4-[4-(2,4-Difluoro-phenyl)-piper...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088845(CHEMBL170307 | N-[4-(4-Phenyl-piperazin-1-ylmethyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088842(CHEMBL171052 | N-{4-[4-(4-Fluoro-phenyl)-piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088843(CHEMBL171115 | N-{4-[4-(4-Methoxy-phenyl)-piperazi...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088847(CHEMBL171345 | N-{4-[4-(4-Chloro-phenyl)-piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of class C beta-lactamase derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088845(CHEMBL170307 | N-[4-(4-Phenyl-piperazin-1-ylmethyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088840(CHEMBL352576 | N-{4-[4-(2,4-Difluoro-phenyl)-piper...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088840(CHEMBL352576 | N-{4-[4-(2,4-Difluoro-phenyl)-piper...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088847(CHEMBL171345 | N-{4-[4-(4-Chloro-phenyl)-piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088847(CHEMBL171345 | N-{4-[4-(4-Chloro-phenyl)-piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50088842(CHEMBL171052 | N-{4-[4-(4-Fluoro-phenyl)-piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105033(CHEMBL112531 | N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)...)
Affinity DataIC50: <0.00100nMAssay Description:In vitro inhibition of [125 I]ET-1 binding to Endothelin A receptor in porcine aortic membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105035(CHEMBL325511 | N-{5-Benzo[1,3]dioxol-5-yl-6-[2-(5-...)
Affinity DataIC50:  0.00110nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50104997(4-tert-Butyl-N-[6-[2-(5-methylsulfanyl-pyrimidin-2...)
Affinity DataIC50:  0.00170nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105034(4-tert-Butyl-N-{6-[2-(5-methoxy-pyrimidin-2-yloxy)...)
Affinity DataIC50:  0.00170nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50107562(CHEMBL168119 | N-[6-[2-(5-Bromo-pyrimidin-2-yloxy)...)
Affinity DataIC50:  0.00250nMAssay Description:In vitro inhibition of [125 I]ET-1 binding to Endothelin A receptor in porcine aortic membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105055(4-tert-Butyl-N-{6-[2-(5-hydroxymethyl-pyrimidin-2-...)
Affinity DataIC50:  0.00260nMAssay Description:Ability to inhibit [125I]ET1 binding to endothelin A receptor in porcine aortic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105048(CHEMBL112144 | N-[6-[2-(5-Bromo-pyrimidin-2-yloxy)...)
Affinity DataIC50:  0.00390nMAssay Description:In vitro inhibition of [125 I]ET-1 binding to Endothelin A receptor in porcine aortic membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tanabe Seiyaku

Curated by ChEMBL
LigandPNGBDBM50105048(CHEMBL112144 | N-[6-[2-(5-Bromo-pyrimidin-2-yloxy)...)
Affinity DataIC50:  0.00390nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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