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Found 71 with Last Name = 'moser' and Initial = 'd'
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50502344(Talinolol)
Affinity DataKi:  240nMAssay Description:Binding affinity to beta1 adrenergic receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50502344(Talinolol)
Affinity DataKi:  900nMAssay Description:Binding affinity to beta2 adrenergic receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50444531(CHEMBL3099680)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant 5-lipoxygenase (unknown origin) expressed in Escherichia coli BL21(DE3) using arachidonic acid as substrate incubated for 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50502345(CHEMBL4566250)
Affinity DataIC50:  77nMAssay Description:Inhibition of recombinant human full length soluble epoxide hydrolase (1 to 555 residues) expressed in Escherichia coli BL21(DE3) using non-fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM25737(12-[(adamantan-1-ylcarbamoyl)amino]dodecanoic acid...)
Affinity DataIC50:  107nMAssay Description:Inhibition of sEH using (3-Phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester) as substrate incubated for 15 mins prior to s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50444531(CHEMBL3099680)
Affinity DataIC50:  170nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50384785(CHEMBL2037376)
Affinity DataIC50:  470nMAssay Description:Inhibition of soluble epoxide hydrolase using (3-Phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester) as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50384786(CHEMBL1364973)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of soluble epoxide hydrolase using (3-Phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester) as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50384782(CHEMBL2037373)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of recombinant 5-lipooxygenase expressed in Escherichia coli BL21 using arachidonic acid as substrate incubated for 15 mins prior to subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50384783(CHEMBL2037374)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of recombinant 5-lipooxygenase expressed in Escherichia coli BL21 using arachidonic acid as substrate incubated for 15 mins prior to subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50502344(Talinolol)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of recombinant human full length soluble epoxide hydrolase (1 to 555 residues) expressed in Escherichia coli BL21(DE3) using non-fluoresce...More data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50444538(CHEMBL1313977)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50394028(CHEMBL2158536)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of sEH using (3-Phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester) as substrate incubated for 15 mins prior to s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50384784(CHEMBL2037375)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of soluble epoxide hydrolase using (3-Phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester) as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50394029(CHEMBL2158537)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of sEH using (3-Phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester) as substrate incubated for 15 mins prior to s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50444532(CHEMBL3099679)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of recombinant 5-lipoxygenase (unknown origin) expressed in Escherichia coli BL21(DE3) using arachidonic acid as substrate incubated for 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50384779(CHEMBL1330331)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of recombinant 5-lipooxygenase expressed in Escherichia coli BL21 using arachidonic acid as substrate incubated for 15 mins prior to subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50444534(CHEMBL3099594)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of recombinant 5-lipoxygenase (unknown origin) expressed in Escherichia coli BL21(DE3) using arachidonic acid as substrate incubated for 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50384781(CHEMBL2037345)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of recombinant 5-lipooxygenase expressed in Escherichia coli BL21 using arachidonic acid as substrate incubated for 15 mins prior to subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50384780(CHEMBL2037372)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of recombinant 5-lipooxygenase expressed in Escherichia coli BL21 using arachidonic acid as substrate incubated for 15 mins prior to subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50444537(CHEMBL3099590)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50384787(CHEMBL2037377)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of soluble epoxide hydrolase using (3-Phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester) as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50394030(CHEMBL2158540)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of sEH using (3-Phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester) as substrate incubated for 15 mins prior to s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50444535(CHEMBL3099592)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of recombinant 5-lipoxygenase (unknown origin) expressed in Escherichia coli BL21(DE3) using arachidonic acid as substrate incubated for 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50384784(CHEMBL2037375)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of recombinant 5-lipooxygenase expressed in Escherichia coli BL21 using arachidonic acid as substrate incubated for 15 mins prior to subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50444539(CHEMBL3099593)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50444537(CHEMBL3099590)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of recombinant 5-lipoxygenase (unknown origin) expressed in Escherichia coli BL21(DE3) using arachidonic acid as substrate incubated for 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50444540(CHEMBL1594316)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50444533(CHEMBL3099678)
Affinity DataIC50:  8.90E+4nMAssay Description:Inhibition of recombinant 5-lipoxygenase (unknown origin) expressed in Escherichia coli BL21(DE3) using arachidonic acid as substrate incubated for 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50078827(2-(pyridin-3-yl)-1H-benzo[d]imidazole | 2-Pyridin-...)
Affinity DataIC50:  9.10E+4nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50444536(CHEMBL3099591)
Affinity DataIC50:  9.10E+4nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50444535(CHEMBL3099592)
Affinity DataIC50:  9.50E+4nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50444532(CHEMBL3099679)
Affinity DataIC50:  1.33E+5nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50180740(2-(furan-2-yl)-1H-benzo[d]imidazole | CHEMBL201094...)
Affinity DataIC50:  2.07E+5nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Goethe University

Curated by ChEMBL
LigandPNGBDBM50444536(CHEMBL3099591)
Affinity DataIC50:  2.37E+5nMAssay Description:Inhibition of recombinant 5-lipoxygenase (unknown origin) expressed in Escherichia coli BL21(DE3) using arachidonic acid as substrate incubated for 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Of Frankfurt

Curated by ChEMBL
LigandPNGBDBM50444533(CHEMBL3099678)
Affinity DataIC50:  3.79E+5nMAssay Description:Inhibition of recombinant soluble epoxide hydrolase (unknown origin) using PHOME as substrate incubated 15 mins prior to substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378608(CHEMBL601721)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378609(CHEMBL601722)
Affinity DataKd:  5.80E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  2.18E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under HBS-EP condition by CM5 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  1.76E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under HEPES condition by CM5 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  1.49E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under NaCl condition by CM5 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  1.78E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under carboxymethyl-dextran sodium salt condition by CM5 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under HBS-EP condition by CM4 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378610(CHEMBL590917)
Affinity DataKd:  2.83E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378611(CHEMBL590827)
Affinity DataKd:  4.44E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378612(CHEMBL394182)
Affinity DataKd:  1.92E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378613(CHEMBL598744)
Affinity DataKd:  1.17E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378614(CHEMBL391051)
Affinity DataKd:  3.39E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378596(CHEMBL609756)
Affinity DataKd:  1.37E+5nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by biocoreMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  800nMAssay Description:Partial agonist activity at recombinant human GAL4-DBD-fused LXRbeta-LBD expressed in HEK293T cells measured after 12 to 14 hrs by dual-glo luciferas...More data for this Ligand-Target Pair
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