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Found 46 with Last Name = 'muench' and Initial = 'd'
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033887(CHEMBL3358611)
Affinity DataKi:  146nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033944(CHEMBL3358598)
Affinity DataKi:  4.77E+3nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033946(CHEMBL3358596)
Affinity DataKi:  6.62E+3nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033888(CHEMBL3358610)
Affinity DataKi:  1.15E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033890(CHEMBL3358608)
Affinity DataKi:  1.24E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033891(CHEMBL3358607)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033892(CHEMBL3358606)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033893(CHEMBL3358605)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033895(CHEMBL3358604)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033896(CHEMBL3358603)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033897(CHEMBL3358602)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033939(CHEMBL3358601)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033940(CHEMBL3358600)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033943(CHEMBL3358599)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033945(CHEMBL3358597)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033947(CHEMBL3358595)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033963(CHEMBL3358594)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033993(CHEMBL3358593)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50034005(CHEMBL3358592)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033889(CHEMBL3358609)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50034007(CHEMBL3358590)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50034008(CHEMBL3358589)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50034006(CHEMBL3358591)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50034080(CHEMBL3358587)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50034036(CHEMBL3358588)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50002363((APH)2-Amino-7-phosphono-heptanoic acid | 2-Amino-...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards AMPA receptor using [3H]AMPA as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004927(4-Phosphonomethyl-piperidine-2-carboxylic acid | 4...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards Ionotropic glutamate receptor kainate using [3H]-kainic acid as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004927(4-Phosphonomethyl-piperidine-2-carboxylic acid | 4...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards AMPA receptor using [3H]AMPA as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50002360((CPP)4-(3-Phosphono-propyl)-piperazine-2-carboxyli...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards Ionotropic glutamate receptor kainate using [3H]-kainic acid as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50010893((R)-2-Amino-4-oxo-5-phosphono-pentanoic acid | 2-A...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards Ionotropic glutamate receptor kainate using [3H]-kainic acid as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004897((APV)2-Amino-5-phosphono-pentanoic acid | (R)-2-Am...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards Ionotropic glutamate receptor kainate using [3H]-kainic acid as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50010893((R)-2-Amino-4-oxo-5-phosphono-pentanoic acid | 2-A...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards AMPA receptor using [3H]AMPA as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004897((APV)2-Amino-5-phosphono-pentanoic acid | (R)-2-Am...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards AMPA receptor using [3H]AMPA as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50002360((CPP)4-(3-Phosphono-propyl)-piperazine-2-carboxyli...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards AMPA receptor using [3H]AMPA as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50002363((APH)2-Amino-7-phosphono-heptanoic acid | 2-Amino-...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards Ionotropic glutamate receptor kainate using [3H]-kainic acid as radioligand; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033887(CHEMBL3358611)
Affinity DataKi:  1.44E+5nMAssay Description:Inhibition of STAT3 (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50213061(CHEMBL2298601)
Affinity DataIC50:  8.60nMAssay Description:Inhibitory activity of the compound against human prostatic Steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50421737(CHEMBL2311174)
Affinity DataIC50: >430nMAssay Description:Inhibitory activity of the compound against human prostatic Steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284139((6aS,8S,10aS,12aS)-8-Hydroxy-1,10a,12a-trimethyl-h...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity of the compound against human prostatic Steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284141((7S,9aR,11aS)-7-Hydroxy-1,9a,11a-trimethyl-hexadec...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity of the compound against human prostatic Steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284137((6aS,10aS,12aS)-1,10a,12a-Trimethyl-hexadecahydro-...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibitory activity of the compound against human prostatic Steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284142((8S,10aR,12aS)-8-Hydroxy-1,10a,12a-trimethyl-3,4,4...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory activity of the compound against human prostatic Steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284138((8R,9aS,11aS)-1,9a,11a-Trimethyl-2-oxo-hexadecahyd...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory activity of the compound against human prostatic Steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284140((6aS,8R,9aS,11aS)-1,9a,11a-Trimethyl-2-oxo-hexadec...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity of the compound against human prostatic Steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033887(CHEMBL3358611)
Affinity DataKd:  287nMAssay Description:Binding affinity to full-length His-tagged STAT3 (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 5B(Homo sapiens (Human))
University Of Toronto Mississauga

Curated by ChEMBL
LigandPNGBDBM50033887(CHEMBL3358611)
Affinity DataKd:  42nMAssay Description:Binding affinity to full-length His-tagged STAT5B (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed