TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of recombinant human Sirt5 incubated for 1 hr by FLUOR DE LYS fluorometric microplate reader assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of recombinant human Sirt5 incubated for 1 hr by FLUOR DE LYS fluorometric microplate reader assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of recombinant human Sirt5 incubated for 1 hr by FLUOR DE LYS fluorometric microplate reader assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of recombinant human Sirt5 incubated for 1 hr by FLUOR DE LYS fluorometric microplate reader assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant human Sirt5 incubated for 1 hr by FLUOR DE LYS fluorometric microplate reader assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataIC50: 2.36E+4nMAssay Description:Inhibition of recombinant human Sirt5 incubated for 1 hr by FLUOR DE LYS fluorometric microplate reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 234nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 9.33E+3nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferens in presence of naloxoneMore data for this Ligand-Target Pair
Affinity DataEC50: 6.16E+3nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 9.33E+3nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferens in presence of naloxoneMore data for this Ligand-Target Pair
Affinity DataEC50: 6.17E+3nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferens in presence of naloxoneMore data for this Ligand-Target Pair
Affinity DataEC50: 575nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferensMore data for this Ligand-Target Pair
TargetMu-type opioid/Nociceptin receptor(Rattus norvegicus (rat))
Bulgarian Academy Of Sciences
Curated by ChEMBL
Bulgarian Academy Of Sciences
Curated by ChEMBL
Affinity DataEC50: 316nMAssay Description:Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Bulgarian Academy Of Sciences
Curated by ChEMBL
Bulgarian Academy Of Sciences
Curated by ChEMBL
Affinity DataEC50: 1.62E+3nMAssay Description:Activity at Wistar rat mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of nal...More data for this Ligand-Target Pair
Affinity DataEC50: 1.66E+3nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of naloxoneMore data for this Ligand-Target Pair
Affinity DataEC50: 6.20nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of naloxoneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Bulgarian Academy Of Sciences
Curated by ChEMBL
Bulgarian Academy Of Sciences
Curated by ChEMBL
Affinity DataEC50: 1.23E+3nMAssay Description:Activity at Wistar rat mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
TargetMu-type opioid/Nociceptin receptor(Rattus norvegicus (rat))
Bulgarian Academy Of Sciences
Curated by ChEMBL
Bulgarian Academy Of Sciences
Curated by ChEMBL
Affinity DataEC50: 550nMAssay Description:Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of...More data for this Ligand-Target Pair
TargetMu-type opioid/Nociceptin receptor(Rattus norvegicus (rat))
Bulgarian Academy Of Sciences
Curated by ChEMBL
Bulgarian Academy Of Sciences
Curated by ChEMBL
Affinity DataEC50: 617nMAssay Description:Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of...More data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.41E+3nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Bulgarian Academy Of Sciences
Curated by ChEMBL
Bulgarian Academy Of Sciences
Curated by ChEMBL
Affinity DataEC50: 1.02E+3nMAssay Description:Activity at Wistar rat mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Bulgarian Academy Of Sciences
Curated by ChEMBL
Bulgarian Academy Of Sciences
Curated by ChEMBL
Affinity DataEC50: 1.15E+3nMAssay Description:Activity at Wistar rat mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of nal...More data for this Ligand-Target Pair
TargetMu-type opioid/Nociceptin receptor(Rattus norvegicus (rat))
Bulgarian Academy Of Sciences
Curated by ChEMBL
Bulgarian Academy Of Sciences
Curated by ChEMBL
Affinity DataEC50: 1.66E+3nMAssay Description:Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataEC50: 8.80E+3nMAssay Description:Binding affinity to Sirt5 in human MCF7 cell lysate by pull down assay based LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Binding affinity to Sirt5 in human MCF7 cell lysate by pull down assay based LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataEC50: 2.57E+4nMAssay Description:Binding affinity to Sirt5 in human MCF7 cell lysate by pull down assay based LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetNucleoside diphosphate kinase, mitochondrial(Homo sapiens)
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataEC50: 4.58E+4nMAssay Description:Binding affinity to NME4 in human MCF7 cell lysate by pull down assay based LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetNucleoside diphosphate kinase, mitochondrial(Homo sapiens)
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataEC50: 7.80E+3nMAssay Description:Binding affinity to NME4 in human MCF7 cell lysate by pull down assay based LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetNucleoside diphosphate kinase, mitochondrial(Homo sapiens)
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataEC50: 1.45E+4nMAssay Description:Binding affinity to NME4 in human MCF7 cell lysate by pull down assay based LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetGlutaryl-CoA dehydrogenase, mitochondrial(Homo sapiens)
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataEC50: 1.73E+4nMAssay Description:Binding affinity to GCDH in human MCF7 cell lysate by pull down assay based LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetGlutaryl-CoA dehydrogenase, mitochondrial(Homo sapiens)
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataEC50: 5.95E+4nMAssay Description:Binding affinity to GCDH in human MCF7 cell lysate by pull down assay based LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 6.17E+3nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 214nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferens in presence of naloxoneMore data for this Ligand-Target Pair
Affinity DataEC50: 407nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferens in presence of naloxoneMore data for this Ligand-Target Pair
TargetGlutaryl-CoA dehydrogenase, mitochondrial(Homo sapiens)
Ludwig-Maximilians University
Curated by ChEMBL
Ludwig-Maximilians University
Curated by ChEMBL
Affinity DataEC50: 5.02E+4nMAssay Description:Binding affinity to GCDH in human MCF7 cell lysate by pull down assay based LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 977nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferens in presence of naloxoneMore data for this Ligand-Target Pair
Affinity DataEC50: 2.34E+3nMAssay Description:Activity against LFES-evoked contraction of Wistar rat vas deferensMore data for this Ligand-Target Pair