Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Relative inhibition of phosphodiesterase 4 activity and Rolipram binding to PDE4More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Binding activity towards Rolipram binding site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of Rolipram binding to phosphodiesterase 4 at 20 uMMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Binding activity towards Rolipram binding site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Binding activity towards Rolipram binding site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:In vitro binding activity towards catalytic site of phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration for half-maximal displacement of 1.0 nM [3H]ADTN specific binding from rat striatal membranes using 10E-5 sulpirideMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration half-maximal displacement of 1.0 nM [3H]NPA specific binding from rat striatal membranes using 10e-5 (+/-)ADTNMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Chiroscience
Curated by ChEMBL
Chiroscience
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding activity towards Rolipram binding site of phosphodiesterase 4More data for this Ligand-Target Pair