Affinity DataKi: 600nMAssay Description:Binding affinity to GFP tagged human mGluR2 containing truncated N-terminal region expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Binding affinity to GFP tagged human mGluR2 containing truncated N-terminal region expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity to GFP tagged human mGluR2 containing truncated N-terminal region expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.60E+3nMAssay Description:Binding affinity to GFP tagged human mGluR2 containing truncated N-terminal region expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Negative allosteric modulator activity at human mGluR2 expressed in HEK cells in presence of glutamate EC80 concentration by Ca2+ functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Negative allosteric modulator activity at human mGluR2 expressed in HEK cells in presence of glutamate EC80 concentration by Ca2+ functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Negative allosteric modulator activity at human mGluR2 expressed in HEK cells in presence of glutamate EC80 concentration by Ca2+ functional assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.84E+4nMAssay Description:Activity at rat mGluR6 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 4.83E+4nMAssay Description:Activity at rat mGluR4 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: >5.00E+6nMAssay Description:Activity at rat mGluR5 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+6nMAssay Description:Activity at rat mGluR2 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+6nMAssay Description:Activity at rat mGluR1 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.34E+4nMAssay Description:Positive allosteric modulator activity at human mGluR3 expressed in HEK cells in presence of glutamate EC10 concentration by Ca2+ functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.90E+3nMAssay Description:Positive allosteric modulator activity at human mGluR3 expressed in HEK cells in presence of glutamate EC10 concentration by Ca2+ functional assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.01E+4nMAssay Description:Activity at rat mGluR8 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat mGluR5 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 5.62E+4nMAssay Description:Activity at rat mGluR8 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.20E+6nMAssay Description:Activity at rat mGluR7 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 7.20E+3nMAssay Description:Activity at rat mGluR4 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.04E+4nMAssay Description:Positive allosteric modulator activity at human mGluR3 expressed in HEK cells in presence of glutamate EC10 concentration by Ca2+ functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat mGluR2 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 3.78E+5nMAssay Description:Activity at rat mGluR6 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair