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Found 816 with Last Name = 'ng' and Initial = 'wl'
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175864(Bz-Nle-Lys-Arg-Arg-B(OH)2 | CHEMBL199845)
Affinity DataKi:  43nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Academia Sinica

LigandPNGBDBM7918(1-(3,4-dimethoxyphenyl)-3-[3-(1H-imidazol-1-yl)pro...)
Affinity DataKi:  95nM ΔG°:  -40.1kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Academia Sinica

LigandPNGBDBM7887(1-Benzylimidazole (BI) | 1-benzyl-1H-imidazole | 1...)
Affinity DataKi:  262nM ΔG°:  -37.6kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Academia Sinica

LigandPNGBDBM7887(1-Benzylimidazole (BI) | 1-benzyl-1H-imidazole | 1...)
Affinity DataKi:  607nM ΔG°:  -35.5kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175863(Bz-Nle-Lys-Arg-Arg-CF3 | CHEMBL200294)
Affinity DataKi:  850nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175982(Bz-Lys-Arg-Arg-H | CHEMBL199510)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Academia Sinica

LigandPNGBDBM7949(Imidazole C-4(5) deriv. 1 | N-[2-(1H-Imidazol-4-yl...)
Affinity DataKi:  1.70E+3nM ΔG°:  -32.9kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Academia Sinica

LigandPNGBDBM7918(1-(3,4-dimethoxyphenyl)-3-[3-(1H-imidazol-1-yl)pro...)
Affinity DataKi:  1.82E+3nM ΔG°:  -32.8kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
TargetKetol-acid reductoisomerase (NADP(+))(Escherichia coli)
Nankai University

LigandPNGBDBM82145(N-hydroxy-N-isopropyloxamate, IpOHA)
Affinity DataKi:  2.75E+3nM ΔG°:  -32.3kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition of E. coli KARI (ketol-acid reductoisomerase) is time dependent, and activity was measured by the decrease in A340 at 30 C in solutions co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175984(BZ-Nle-Lys-Arg-(4-guanidinyl)-Phe-H | Bz-Nle-Lys-A...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175976(Bz-Ala-Lys-Arg-Arg-H | CHEMBL197765)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Academia Sinica

LigandPNGBDBM7949(Imidazole C-4(5) deriv. 1 | N-[2-(1H-Imidazol-4-yl...)
Affinity DataKi:  5.75E+3nM ΔG°:  -29.9kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM33259(Bz-NKRR-H | Bz-Nle-Lys-Arg-Arg-H | CHEMBL256877)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM33259(Bz-NKRR-H | Bz-Nle-Lys-Arg-Arg-H | CHEMBL256877)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175988(Bz-Nle-Lys-Arg-(p-Me)Phe-H | CHEMBL199396)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175987(Bz-Phe-Lys-Arg-Arg-H | CHEMBL199736)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175974(Bz-Nle-Lys-Arg-Trp-H | CHEMBL433993)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175993(Bz-D-Nle-Lys-Arg-Arg-H | CHEMBL201775)
Affinity DataKi:  9.40E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175978(Bz-Nle-Lys-Arg-(p-Ph)Phe-H | CHEMBL381854)
Affinity DataKi:  1.16E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175981(Bz-Arg-Arg-H | CHEMBL197766)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175985(Bz-Nle-Phe-Arg-Arg-H | CHEMBL199582)
Affinity DataKi:  1.58E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175986(Bz-Nle-Lys-Arg-Phe-H | CHEMBL199727)
Affinity DataKi:  1.59E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175968(Bz-Nle-Lys-Arg-(p-CN)Phe-H | CHEMBL200095)
Affinity DataKi:  1.86E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175971(Bz-Nle-Lys-Arg-Lys-H | CHEMBL377076)
Affinity DataKi:  2.05E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175970(Bz-Nle-Ala-Arg-Arg-H | CHEMBL369916)
Affinity DataKi:  2.21E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175975(Bz-Nle-D-Lys-Arg-Arg-H | CHEMBL370138)
Affinity DataKi:  2.86E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKetol-acid reductoisomerase (NADP(+))(Escherichia coli)
Nankai University

LigandPNGBDBM82144(Cyclopropane, 5)
Affinity DataKi:  3.12E+4nM ΔG°:  -26.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition of E. coli KARI (ketol-acid reductoisomerase) is time dependent, and activity was measured by the decrease in A340 at 30 C in solutions co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175991(Bz-Nle-Lys-Arg-Phg-H | CHEMBL200972)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175990(Bz-Nle-Lys-Phe-Arg-H | CHEMBL435122)
Affinity DataKi:  4.07E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175977(Bz-Nle-Lys-Lys-Arg-H | CHEMBL201609)
Affinity DataKi:  4.13E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50228800(Bz-Nle-Lys-Arg-Arg-Thiazole | CHEMBL271094 | N-((S...)
Affinity DataKi:  4.28E+4nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175969(Bz-N-Me-Nle-Lys-Arg-Arg-H | CHEMBL382143)
Affinity DataKi:  4.37E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175967(Bz-Nle-Lys-N-Me-Arg-Arg-H | CHEMBL199726)
Affinity DataKi:  4.74E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175980(Bz-Nle-Lys-Arg-D-Arg-H | CHEMBL199352)
Affinity DataKi:  5.10E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175979(Bz-Nle-Pro-Arg-Arg-H | CHEMBL382983)
Affinity DataKi:  6.14E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKetol-acid reductoisomerase (NADP(+))(Escherichia coli)
Nankai University

LigandPNGBDBM82142(Cyclopropane, 3)
Affinity DataKi:  7.66E+4nM ΔG°:  -23.9kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition of E. coli KARI (ketol-acid reductoisomerase) is time dependent, and activity was measured by the decrease in A340 at 30 C in solutions co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50228798(Bz-Nle-Lys-Arg-Arg-Benzoxazole | CHEMBL256870 | N-...)
Affinity DataKi:  8.29E+4nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKetol-acid reductoisomerase (NADP(+))(Escherichia coli)
Nankai University

LigandPNGBDBM82143(Cyclopropane, 4)
Affinity DataKi:  9.53E+4nM ΔG°:  -23.3kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition of E. coli KARI (ketol-acid reductoisomerase) is time dependent, and activity was measured by the decrease in A340 at 30 C in solutions co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175965(Bz-Nle-Lys-Pro-Arg-H | CHEMBL199987)
Affinity DataKi:  1.09E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175973(Bz-Nle-N-Me-Lys-Arg-Arg-H | CHEMBL381639)
Affinity DataKi:  1.13E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175989(Bz-Nle-Lys-D-Arg-Arg-H | CHEMBL371447)
Affinity DataKi:  1.15E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175869(Bz-Nle-Lys-Arg-Arg-NH2 | CHEMBL198384)
Affinity DataKi:  1.28E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175972(Bz-Nle-Lys-Arg-(p-Cl)Phe-H | CHEMBL199531)
Affinity DataKi:  1.38E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175865(Bz-Nle-Lys-Arg-Arg(OH)-CONH-Bn | CHEMBL369918)
Affinity DataKi:  1.78E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175966(Bz-Nle-Lys-Arg-Ala-H | CHEMBL199376)
Affinity DataKi:  1.93E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175860(Bz-Nle-Lys-Thr-Arg-OH | CHEMBL383351)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175862(Bz-Nle-Lys-Arg-Arg-H | Bz-Nle-Lys-Arg-Arg-OH | CHE...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175992(Bz-Nle-Lys-Arg-homoPhe-H | CHEMBL370338)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175858(Bz-Nle-Lys-Arg-Arg-NHSO2CF3 | CHEMBL369917)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50175983(Bz-Nle-Lys-Ala-Arg-H | CHEMBL372963)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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