TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity towards dopamine transporter using [3H]WIN-35428 as radioligand from rat caudate putamen tissue (high affinity)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity towards dopamine transporter using [3H]WIN-35428 as radioligand from rat caudate putamen tissue (high affinity)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Binding affinity towards dopamine transporter using [3H]WIN-35428 as radioligand from rat caudate putamen tissue (high affinity)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataKi: 124nMAssay Description:Binding affinity towards dopamine transporter using [3H]WIN-35428 as radioligand from rat caudate putamen tissue (low affinity for one set model)More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataKi: 224nMAssay Description:Binding affinity towards dopamine transporter using [3H]WIN-35428 as radioligand from rat caudate putamen tissue (low affinity)More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataKi: 314nMAssay Description:Binding affinity towards dopamine transporter using [3H]WIN-35428 as radioligand from rat caudate putamen tissue (low affinity)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataKi: 388nMAssay Description:Binding affinity towards dopamine transporter using [3H]WIN-35428 as radioligand from rat caudate putamen tissue (low affinity)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of New Orleans
Curated by ChEMBL
University Of New Orleans
Curated by ChEMBL
Affinity DataKi: 2.28E+3nMAssay Description:Binding affinity towards dopamine transporter using [3H]WIN-35428 as radioligand from rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
The Ohio State University
Curated by ChEMBL
The Ohio State University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human ERG expressed in CHOK1 cells by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma
Curated by ChEMBL
Purdue Pharma
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Antagonist activity in capsaicin-induced FLIPR assays in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase using relaxed pBR322 as substrate by gel electrophoresisMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity incubated for 25 min by ethidium bromide/bromophenol blue staining based agarose...More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase using relaxed pBR322 as substrate by gel electrophoresisMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma
Curated by ChEMBL
Purdue Pharma
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Antagonist activity in capsaicin-induced FLIPR assays in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma
Curated by ChEMBL
Purdue Pharma
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Antagonist activity in capsaicin-induced FLIPR assays in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pBR322 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma
Curated by ChEMBL
Purdue Pharma
Curated by ChEMBL
Affinity DataIC50: 104nMpH: 5.5Assay Description:Antagonist activity in pH 5.5-induced FLIPR assays in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma
Curated by ChEMBL
Purdue Pharma
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Antagonist activity in capsaicin-induced FLIPR assays in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of Staphylococcus aureus Gyrase supercoiling activity assessed as reduction in supercoiling pBR322 DNA by measuring relaxation by bromophe...More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase using relaxed pBR322 as substrate by gel electrophoresisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma
Curated by ChEMBL
Purdue Pharma
Curated by ChEMBL
Affinity DataIC50: 136nMAssay Description:Antagonist activity in capsaicin-induced FLIPR assays in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair