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Found 28 with Last Name = 'novello' and Initial = 'pm'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335534(1-(1-benzylpiperidin-4-yl)-3-(pyridin-3-yl)thioure...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335534(1-(1-benzylpiperidin-4-yl)-3-(pyridin-3-yl)thioure...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335534(1-(1-benzylpiperidin-4-yl)-3-(pyridin-3-yl)thioure...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335543(1-(2-phenoxyethyl)-3-(2-(piperidin-1-yl)ethyl)-1H-...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335541(4,6,8-trimethyl-N-(4,4,6-trimethyl-1,4-dihydropyri...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335542(2-(2-(3H-indol-3-ylidene)ethylidene)-1-methyl-1,2-...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335540(3-Methoxy-5-(3-methylthio-1,2,4-triazin-5-yl-)-1,2...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335547(7-ethoxy-4-methyl-N-(4,4,6-trimethyl-4,5-dihydropy...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335546(7-ethyl-4-methyl-N-(4,4,6-trimethyl-4,5-dihydropyr...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50313985(8-methyl-8-azabicyclo[3.2.1]octan-3-one O-(4-chlor...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335535(1-(1-benzylpiperidin-4-yl)-3-phenylthiourea | CHEM...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335539(3-cyanoquinuclidin-3-yl acetate | CHEMBL1652416)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335545(3-(methylthio)-5-phenyl-1,2,4-triazine | CHEMBL136...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335544(1-(methylthio)-4-(3-(methylthio)-1,2,4-triazin-5-y...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335538(1-(1-ethylpiperidin-4-yl)-3-(pyridin-3-yl)thiourea...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335537(1-(1-benzylpiperidin-4-yl)-3-(pyridin-3-yl)urea | ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335536(1-(1-benzylpiperidin-4-yl)-3-propylthiourea | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50201554(1-benzyl-3-(2-(2-(2-(3-benzyl-2-imino-2,3-dihydrob...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human glutathione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50201552(1-(3,4-dichlorophenyl)-2-(2-imino-3-(2-(piperidin-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human glutathione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50201545(1-(3,4-dichlorophenyl)-2-(3-(2-(dimethylamino)ethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human glutathione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335548(5,6-dimethyl-2-(4,6,8-trimethylquinazolin-2-ylamin...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335549(CHEMBL1652425 | N-(4,6-dimethylpyrimidin-2-yl)-4,5...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335550(CHEMBL1652426 | N-(4,6-dimethylpyrimidin-2-yl)-4,6...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335551(1-(4,6,8-trimethylquinazolin-2-yl)guanidine | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335552(1-(4-methylquinazolin-2-yl)guanidine | CHEMBL60236...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 trypanothione reductase assessed as inhibition of thionitrobenzoate formation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50335543(1-(2-phenoxyethyl)-3-(2-(piperidin-1-yl)ethyl)-1H-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50313985(8-methyl-8-azabicyclo[3.2.1]octan-3-one O-(4-chlor...)
Affinity DataEC50:  3.50E+4nMAssay Description:Inhibition of Trypanosoma cruzi X10/1 recombinant trypanoythione reductase assessed as increase in absorbance at 410 nm due to the formation of TNBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed