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Found 26 with Last Name = 'oatis' and Initial = 'je'
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM50008781(7-(3-(2-ethyl-N-phenylhydrazinecarboxamide)-7-oxa-...)
Affinity DataKi:  4.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM81948(CAS_89617-02-7 | ONO 11,113 | ONO-11113 | STA2)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM81949(9,11-AzoPGH2 | 9,11-azo PGH2 | J389.306E | PGH2, 9...)
Affinity DataKi:  41nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM50018531((Z)-7-[(S)-6-((E)-(S)-3-Hydroxy-oct-1-enyl)-2-oxa-...)
Affinity DataKi:  62nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM81947(CAS_113243-00-8 | L-657926)
Affinity DataKi:  424nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM81947(CAS_113243-00-8 | L-657926)
Affinity DataIC50:  11nMAssay Description:Binding affinity towards Thromboxane A2/ Prostaglandin H2 receptor in human platelet membranes using [125I]- as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM81947(CAS_113243-00-8 | L-657926)
Affinity DataIC50:  11.2nMAssay Description:Binding affinity towards Thromboxane A2/ Prostaglandin H2 receptor in human platelet membranes using [125I]- as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50050098((S)-Phenyl-(S)-piperidin-2-yl-acetic acid methyl e...)
Affinity DataIC50:  19.9nMAssay Description:Inhibition of [3H]dopamine uptake in HEK293 cells expressing human dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM50452544(CHEMBL2448578)
Affinity DataIC50:  36nMAssay Description:Binding affinity towards Thromboxane A2 receptor/Prostaglandin receptor in human platelet membranes using [125I]- as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM82512(CAS_128719-90-4 | I-BOP)
Affinity DataIC50:  50nMAssay Description:Binding affinity towards Thromboxane A2 receptor/Prostaglandin receptor in human platelet membranes using [125I]- as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50050098((S)-Phenyl-(S)-piperidin-2-yl-acetic acid methyl e...)
Affinity DataIC50:  51nMAssay Description:Inhibition of [3H]norepinephrine uptake in HEK293 cells expressing human norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50165211((2R,2'R)-Phenyl-piperidin-2-yl-acetic acid ethyl e...)
Affinity DataIC50:  95nMAssay Description:Inhibition of [3H]dopamine uptake in HEK293 cells expressing human dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50050098((S)-Phenyl-(S)-piperidin-2-yl-acetic acid methyl e...)
Affinity DataIC50:  122nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  289nMAssay Description:Inhibition of [3H]5-HT uptake in HEK293 cells expressing human serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  289nMAssay Description:Inhibition of [3H]dopamine uptake in HEK293 cells expressing human dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50165211((2R,2'R)-Phenyl-piperidin-2-yl-acetic acid ethyl e...)
Affinity DataIC50:  319nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  367nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  433nMAssay Description:Displacement of [125I]RTI-55 from human Serotonin transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  462nMAssay Description:Inhibition of [3H]norepinephrine uptake in HEK293 cells expressing human norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50165211((2R,2'R)-Phenyl-piperidin-2-yl-acetic acid ethyl e...)
Affinity DataIC50:  480nMAssay Description:Inhibition of [3H]norepinephrine uptake in HEK293 cells expressing human norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50050098((S)-Phenyl-(S)-piperidin-2-yl-acetic acid methyl e...)
Affinity DataIC50:  788nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  2.99E+3nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50165211((2R,2'R)-Phenyl-piperidin-2-yl-acetic acid ethyl e...)
Affinity DataIC50: >7.20E+3nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50165211((2R,2'R)-Phenyl-piperidin-2-yl-acetic acid ethyl e...)
Affinity DataIC50:  7.54E+3nMAssay Description:Displacement of [125I]RTI-55 from human Serotonin transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50165211((2R,2'R)-Phenyl-piperidin-2-yl-acetic acid ethyl e...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]5-HT uptake in HEK293 cells expressing human serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50050098((S)-Phenyl-(S)-piperidin-2-yl-acetic acid methyl e...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]RTI-55 from human Serotonin transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed