TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 92nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory concentration against blocking of E-selectin during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory concentration against blocking of Selectin P during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibitory concentration against blocking of Selectin P during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibitory concentration against blocking of Selectin P during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+5nMAssay Description:Inhibitory concentration against blocking of E-selectin during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+5nMAssay Description:Inhibitory concentration against blocking of E-selectin during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against blocking of Selectin P during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against blocking of E-selectin during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 1.90nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 6.70nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 53nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataKd: 0.110nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataKd: 0.800nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataKd: 0.410nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataKd: 0.640nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataKd: 0.400nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataKd: 1.80nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataKd: 0.100nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataKd: 2.90nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 3.60nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 2.20nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 6.70nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 2.20nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataKd: 1.10E+5nMAssay Description:Binding affinity to PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at human PPARalpha assessed as transactivation activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 43nMAssay Description:Agonist activity at human PPARdelta assessed as transactivation activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 54nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 840nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 0.720nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 620nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair