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Found 85 with Last Name = 'ohashi' and Initial = 'm'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50492981(CHEMBL2413327)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50492983(CHEMBL2413333)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50492978(CHEMBL2413228)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50492980(CHEMBL2413324)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50492982(CHEMBL2413325)
Affinity DataIC50:  92nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50492979(CHEMBL2413326)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50266373(2-chloro-5-nitro-N-(pyridin-4-yl)benzamide | CHEMB...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human PPARdelta assessed as effect on TIPP-703-induced activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50050500(CHEMBL3085443 | Sodium; 3,5-dihydroxy-2-[5-hydroxy...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory concentration against blocking of E-selectin during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50050500(CHEMBL3085443 | Sodium; 3,5-dihydroxy-2-[5-hydroxy...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory concentration against blocking of Selectin P during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50050500(CHEMBL3085443 | Sodium; 3,5-dihydroxy-2-[5-hydroxy...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50422136(CHEMBL2303852)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50422136(CHEMBL2303852)
Affinity DataIC50:  2.50E+5nMAssay Description:Inhibitory concentration against blocking of Selectin P during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50050501(CHEMBL60263 | Sodium; 3,5-dihydroxy-2-[5-hydroxy-2...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibitory concentration against blocking of Selectin P during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50422136(CHEMBL2303852)
Affinity DataIC50:  3.30E+5nMAssay Description:Inhibitory concentration against blocking of E-selectin during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50450369(SIALYL LEWIS X | Sialyl LeX | Sialyl lewis-x | sLe...)
Affinity DataIC50:  6.00E+5nMAssay Description:Inhibitory concentration against blocking of E-selectin during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50050501(CHEMBL60263 | Sodium; 3,5-dihydroxy-2-[5-hydroxy-2...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50450369(SIALYL LEWIS X | Sialyl LeX | Sialyl lewis-x | sLe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against blocking of Selectin P during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50450369(SIALYL LEWIS X | Sialyl LeX | Sialyl lewis-x | sLe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
New Drug Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50050501(CHEMBL60263 | Sodium; 3,5-dihydroxy-2-[5-hydroxy-2...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against blocking of E-selectin during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050556(CHEMBL3317860)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050560(CHEMBL3317859)
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050557(CHEMBL3317858)
Affinity DataEC50:  53nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050550(CHEMBL3317867)
Affinity DataKd:  0.110nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050551(CHEMBL3317866)
Affinity DataKd:  0.800nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050552(CHEMBL3317865)
Affinity DataKd:  0.410nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050553(CHEMBL3317864)
Affinity DataKd:  0.640nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050554(CHEMBL3317863)
Affinity DataKd:  0.400nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050555(CHEMBL3317455)
Affinity DataKd:  1.80nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050556(CHEMBL3317860)
Affinity DataKd:  0.100nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050557(CHEMBL3317858)
Affinity DataKd:  2.90nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50335272((R)-2-Benzyl-3-(3-(((4-adamantan-1-yl)benzamido)-m...)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050550(CHEMBL3317867)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050551(CHEMBL3317866)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050552(CHEMBL3317865)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050553(CHEMBL3317864)
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050554(CHEMBL3317863)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050558(CHEMBL3317862)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050559(CHEMBL3317861)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050555(CHEMBL3317455)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM19264((4E)-6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1,3-dih...)
Affinity DataKd:  1.10E+5nMAssay Description:Binding affinity to PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50365345(CHEMBL1956149)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PPARalpha assessed as transactivation activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50365345(CHEMBL1956149)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human PPARdelta assessed as transactivation activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50231507((2S)-2-(4-propoxy-3-{[({4-[(3S,5S,7S)-tricyclo[3.3...)
Affinity DataEC50:  54nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50176605((S)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  12nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50176605((S)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  23nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50176609((R)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  150nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50176609((R)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  840nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50214207((2S)-2-{4-butoxy-3-[({[2-fluoro-4-(trifluoromethyl...)
Affinity DataEC50:  250nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50214207((2S)-2-{4-butoxy-3-[({[2-fluoro-4-(trifluoromethyl...)
Affinity DataEC50:  0.720nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50214209((R)-2-(4-butoxy-3-((2-fluoro-4-(trifluoromethyl)be...)
Affinity DataEC50:  620nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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