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Found 3035 with Last Name = 'or' and Initial = 'ys'
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008382(Ac-Phe-Lys-AspMet-GIn-Leu-Gly-Arg-OH | CHEMBL23706...)
Affinity DataKi:  200nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008383(CHEMBL408929 | H-Ala-Asn-Ile-Ser-Phe-Lys-AspMet-GI...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008377(CHEMBL132959 | H-Phe-Lys-AspMet-GIn-Leu-Gly-Arg-OH)
Affinity DataKi:  260nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008381(CHEMBL441393 | H-Ile-Ser-Phe-Lys-AspMet-GIn-Leu-Gl...)
Affinity DataKi:  390nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50405349(CHEMBL5271837)
Affinity DataKi:  740nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405333(CHEMBL5270570)
Affinity DataKi:  744nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008373(CHEMBL439468 | H-Leu-Arg-Ala-Asn-Ile-Ser-Phe-Lys-A...)
Affinity DataKi:  810nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50229889(CHEMBL3350366)
Affinity DataKi:  1.60E+3nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008231(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  2.00E+3nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008371(CHEMBL127385 | H-Thi-Lys-AspMet-GIn-Leu-Gly-Arg-OH)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008230(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  2.90E+3nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50405348(CHEMBL5280643)
Affinity DataKi:  3.00E+3nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008374(CHEMBL435002 | Hca-Lys-AspMet-GIn-Leu-Gly-Arg-OH)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008233(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  5.30E+3nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008232(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  1.00E+4nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008379(CHEMBL339127 | H-Cha-Lys-AspMet-GIn-Leu-Gly-Arg-OH)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008375(CHEMBL128360 | H-Thia-Lys-AspMet-GIn-Leu-Gly-Arg-O...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008228(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  2.50E+4nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008372(CHEMBL408493 | H-Phg-Lys-AspMet-GIn-Leu-Gly-Arg-OH)
Affinity DataKi:  3.10E+4nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008380(CHEMBL217002 | H-hPhe-Lys-AspMet-GIn-Leu-Gly-Arg-O...)
Affinity DataKi:  3.60E+4nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008384(CHEMBL336081 | H-His(3Me)-Lys-AspMet-GIn-Leu-Gly-A...)
Affinity DataKi:  5.80E+4nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008370(CHEMBL435810 | H-DPhe-Lys-AspMet-GIn-Leu-Gly-Arg-O...)
Affinity DataKi:  7.90E+4nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50405346(CHEMBL5266306)
Affinity DataKi:  8.50E+4nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405336(CHEMBL5277116)
Affinity DataKi:  1.39E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008235(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  1.50E+5nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50405334(CHEMBL5280829)
Affinity DataKi:  1.55E+5nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405329(CHEMBL5279025)
Affinity DataKi:  1.74E+5nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced platelet aggregation in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008378(CHEMBL129978 | H-His(1Me)-Lys-AspMet-GIn-Leu-Gly-A...)
Affinity DataKi:  1.80E+5nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008226(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  2.10E+5nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008376(2-[2-(2-{2-[2-(2-{6-Amino-2-[2-amino-3-(3H-imidazo...)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50405337(CHEMBL5268186)
Affinity DataKi:  3.54E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405328(CHEMBL5278563)
Affinity DataKi:  3.90E+5nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced platelet aggregation in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405341(CHEMBL5287370)
Affinity DataKi:  5.40E+5nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405343(CHEMBL5279009)
Affinity DataKi:  5.88E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008229(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  6.00E+5nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008227(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  7.50E+5nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50405340(CHEMBL5276693)
Affinity DataKi:  9.55E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405347(CHEMBL5281989)
Affinity DataKi:  1.42E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405342(CHEMBL5273882)
Affinity DataKi:  2.10E+6nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405344(CHEMBL5278260)
Affinity DataKi:  4.74E+6nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405338(CHEMBL2393369)
Affinity DataKi:  5.00E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405331(CHEMBL5276685)
Affinity DataKi:  5.00E+6nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced platelet aggregation in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405339(CHEMBL5286003)
Affinity DataKi:  6.22E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405345(CHEMBL5273503)
Affinity DataKi:  6.38E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405332(CHEMBL5285449)
Affinity DataKi:  1.00E+7nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405335(CHEMBL2357735)
Affinity DataKi:  2.00E+7nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM555177(US11339170, Example 1 | US11339170, Example 2)
Affinity DataIC50: <0.100nMAssay Description:SARS-CoV-2 3C-like (3CL) protease fluorescence assay (FRET): Recombinant SARS-CoV-2 3CL-protease was expressed and purified. TAMRA-SITSAVLQSGFRKMIK-D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReplicase polyprotein 1ab(2019-nCoV)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM555177(US11339170, Example 1 | US11339170, Example 2)
Affinity DataIC50: <0.100nMAssay Description:SARS-CoV-2 3C-like (3CL) protease fluorescence assay (FRET): Recombinant SARS-CoV-2 3CL-protease was expressed and purified. TAMRA-SITSAVLQSGFRKMIK-D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReplicase polyprotein 1ab(2019-nCoV)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM555237(US11339170, Example 72)
Affinity DataIC50: <0.100nMAssay Description:SARS-CoV-2 3C-like (3CL) protease fluorescence assay (FRET): Recombinant SARS-CoV-2 3CL-protease was expressed and purified. TAMRA-SITSAVLQSGFRKMIK-D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReplicase polyprotein 1ab(2019-nCoV)
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM555236(US11339170, Example 71)
Affinity DataIC50: <0.100nMAssay Description:SARS-CoV-2 3C-like (3CL) protease fluorescence assay (FRET): Recombinant SARS-CoV-2 3CL-protease was expressed and purified. TAMRA-SITSAVLQSGFRKMIK-D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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