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Found 449 with Last Name = 'osman' and Initial = 'h'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50614417(CHEMBL4647601)
Affinity DataKi:  0.0500nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50614416(CHEMBL120225)
Affinity DataKi:  4nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50479982(Aptivus | CHEBI:63628 | Tipranavir | U-140690 | US...)
Affinity DataKi:  8nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50614415(CHEMBL5266669)
Affinity DataKi:  15nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM770(4-hydroxy-6-(1-phenylbutan-2-yl)-3-(1-phenylpropyl...)
Affinity DataKi:  38nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM1934(3-[cyclopropyl(phenyl)methyl]-4-hydroxy-7-methoxy-...)
Affinity DataKi:  170nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM1932(3-[cyclopropyl(phenyl)methyl]-4-hydroxy-2H-chromen...)
Affinity DataKi:  350nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM1930(4-hydroxy-7-methoxy-3-(1-phenylpropyl)-2H-chromen-...)
Affinity DataKi:  560nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50447970(CHEMBL3115043)
Affinity DataKi:  6.76E+3nMAssay Description:Mixed-type inhibition of equine serum BChE using S-butyrylthiocholine chloride as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50614424(CHEMBL478728)
Affinity DataIC50:  0.0100nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)TBA
LigandPNGBDBM50029982(12-Hydroxy-6,6,10,11-tetramethyl-4-phenyl-11,12-di...)
Affinity DataIC50:  38nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50360916(CHEMBL1935151)
Affinity DataIC50:  110nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Madurai Kamaraj University

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  120nMAssay Description:Inhibition of AChE (unknown origin) using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured every minute by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Madurai Kamaraj University

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  120nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  120nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)TBA
LigandPNGBDBM50029987(12-Hydroxy-6,6,10,11-tetramethyl-4-phenyl-11,12-di...)
Affinity DataIC50:  130nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM2572(2-(4-{4-hydroxy-2-oxo-3-[(2-phenylethyl)sulfanyl]-...)
Affinity DataIC50:  160nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM2509((+/-)-3-[Cyclopentyl(cyclopentylthio)methyl]-4-hyd...)
Affinity DataIC50:  225nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50360911(CHEMBL1935146)
Affinity DataIC50:  340nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50360906(CHEMBL1935141)
Affinity DataIC50:  480nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM993(4,7-dihydroxy-3-[4-(2-methoxyphenyl)butyl]-2H-chro...)
Affinity DataIC50:  520nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50445716(CHEMBL3104317)
Affinity DataIC50:  530nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50346981(CHEMBL1795895)
Affinity DataIC50:  720nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Madurai Kamaraj University

Curated by ChEMBL
LigandPNGBDBM50242974(CHEMBL4072825)
Affinity DataIC50:  780nMAssay Description:Inhibition of AChE (unknown origin) using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured every minute by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50445693(CHEMBL3104448)
Affinity DataIC50:  800nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434513(CHEMBL2385778)
Affinity DataIC50:  800nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50439104(CHEMBL2417659)
Affinity DataIC50:  920nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Madurai Kamaraj University

Curated by ChEMBL
LigandPNGBDBM50558500(CHEMBL4752440)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate preincubated with enzyme for 15 mins followed by substrate addition...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50360907(CHEMBL1935142)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50360917(CHEMBL1935152)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Madurai Kamaraj University

Curated by ChEMBL
LigandPNGBDBM50558514(CHEMBL4747183)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate preincubated with enzyme for 15 mins followed by substrate addition...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434513(CHEMBL2385778)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50445693(CHEMBL3104448)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50346977(CHEMBL1795891)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50439097(CHEMBL1987383)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434506(CHEMBL2385785)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50445719(CHEMBL3104452)
Affinity DataIC50:  1.47E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50360912(CHEMBL1935147)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50445715(CHEMBL3104318)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434511(CHEMBL2385780)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50008529(CHEMBL3235940)
Affinity DataIC50:  1.68E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50445716(CHEMBL3104317)
Affinity DataIC50:  1.71E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50445719(CHEMBL3104452)
Affinity DataIC50:  1.74E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50439093(CHEMBL2417668)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of horse serum BChE using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50614418(CHEMBL5271554)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50614423(CHEMBL5284565)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50445718(CHEMBL3104453)
Affinity DataIC50:  2.05E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50008675(CHEMBL3235947)
Affinity DataIC50:  2.07E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50439096(CHEMBL2417665)
Affinity DataIC50:  2.07E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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