Affinity DataKi: 0.0500nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 8nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 38nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 6.76E+3nMAssay Description:Mixed-type inhibition of equine serum BChE using S-butyrylthiocholine chloride as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 38nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of AChE (unknown origin) using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured every minute by...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 225nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Inhibition of AChE (unknown origin) using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured every minute by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate preincubated with enzyme for 15 mins followed by substrate addition...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate preincubated with enzyme for 15 mins followed by substrate addition...More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine as substrate measured every sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of horse serum BChE using S-butyrylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand Info
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of Electrophorus electricus acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair