Affinity DataKi: 0.130nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]-DAGO) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]-DAGO) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]-DAGO) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 187nMAssay Description:In vitro binding activity against opioid receptor delta using [3DPDPE] as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 809nMAssay Description:In vitro binding activity against opioid receptor delta using [3H]-DPDPE) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]-DAGO) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]-DAGO) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro binding activity against opioid receptor delta using [3H]-DPDPE) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.89E+3nMAssay Description:In vitro binding activity against opioid receptor kappa using [3H]-EKC as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding activity against opioid receptor kappa using [3H]-EKC) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding activity against opioid receptor kappa using [3H]-EKC) as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding activity against opioid receptor kappa using [3H]-EKC) as radioligandMore data for this Ligand-Target Pair