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Found 196 with Last Name = 'osterkamp' and Initial = 'f'
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217428(2S,3R,5S-4-{[2-carboxy-2-(2,4,6-trimethyl-benzoyla...)
Affinity DataIC50:  0.540nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217419(2S,3R,5S-3-(2-{1-(3,3-dimethyl-butyryl)-5-[(4-meth...)
Affinity DataIC50:  0.550nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217426(2S,3R,5S-3-(2-{1-(3,3-dimethyl-butyryl)-5-[(4-meth...)
Affinity DataIC50:  0.550nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217425(2S,3R,5S-4-({2-carboxy-2-[(1-methyl-cyclohexanecar...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466499(US10799605, Example 4)
Affinity DataIC50:  0.870nMAssay Description:In order to determine the binding affinity of compounds comprising a radiolabel for NTR1, a radioligand binding assay was carried out. A radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423732(CHEMBL590389)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217422(2S,3R,20S-3-(2-{1-(3,3-dimethyl-butyryl)-5-[(4-met...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423736(CHEMBL591543)
Affinity DataIC50:  0.920nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217435(2S,4R,20S-4-{[2-carboxy-2-(2,4,6-trimethyl-benzene...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217427(2S,3R,5S-3-{2-[1-(3,3-dimethyl-butyryl)-5-(pyridin...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423726(CHEMBL594161)
Affinity DataIC50:  1.5nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217432(2S,3R,5S-3-{2-[1-(3,3-dimethyl-butyryl)-5-(pyridin...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423717(CHEMBL594166)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423737(CHEMBL591544)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423728(CHEMBL593938)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217423(2S,4R,20S-4-({2-carboxy-2-[(1-methyl-cyclohexaneca...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423731(CHEMBL590622)
Affinity DataIC50:  2nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423735(CHEMBL592769)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423738(CHEMBL591545)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217435(2S,4R,20S-4-{[2-carboxy-2-(2,4,6-trimethyl-benzene...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of integrin alphaVbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423718(CHEMBL606371)
Affinity DataIC50:  2.5nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423739(CHEMBL591778)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466500(US10799605, Example 5)
Affinity DataIC50:  2.90nMAssay Description:In order to determine the binding affinity of compounds comprising a radiolabel for NTR1, a radioligand binding assay was carried out. A radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466502(US10799605, Example 13)
Affinity DataIC50:  3nMAssay Description:In order to determine the binding affinity of compounds comprising a radiolabel for NTR1, a radioligand binding assay was carried out. A radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466505(US10799605, Example 19)
Affinity DataIC50:  3.40nMAssay Description:In order to determine the binding affinity of compounds comprising a radiolabel for NTR1, a radioligand binding assay was carried out. A radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217434(2S,4R,20S-4-{[2-carboxy-2-(2,4,6-trimethyl-benzoyl...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217420(12S,14R,30S-4-{[2-carboxy-2-(2,4,6-trimethylbenzen...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217422(2S,3R,20S-3-(2-{1-(3,3-dimethyl-butyryl)-5-[(4-met...)
Affinity DataIC50:  4nMAssay Description:Inhibition of integrin alphaVbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423733(CHEMBL599877)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466501(US10799605, Example 12)
Affinity DataIC50:  4.90nMAssay Description:In order to determine the binding affinity of compounds comprising a radiolabel for NTR1, a radioligand binding assay was carried out. A radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466504(US10799605, Example 18)
Affinity DataIC50:  5.30nMAssay Description:In order to determine the binding affinity of compounds comprising a radiolabel for NTR1, a radioligand binding assay was carried out. A radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217430(2S,3R,5S-3-{2-[1-(3,3-dimethylbutyryl)-5-(pyridin-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423724(CHEMBL596248)
Affinity DataIC50:  6.10nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217431(2S,4R,20S-4-[(2-benzenesulfonylamino-2-carboxy-eth...)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of integrin alphaVbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466499(US10799605, Example 4)
Affinity DataIC50:  7.54nMAssay Description:Ca2+ ions are usually kept at nanomolar levels in the cytosol of cells, and act in a number of signal transduction pathways as second messengers. Man...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217435(2S,4R,20S-4-{[2-carboxy-2-(2,4,6-trimethyl-benzene...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466504(US10799605, Example 18)
Affinity DataIC50:  8.95nMAssay Description:Ca2+ ions are usually kept at nanomolar levels in the cytosol of cells, and act in a number of signal transduction pathways as second messengers. Man...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217421((S)-3-(2-((3R,5S)-1-(methoxycarbonyl)-5-((pyridin-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of integrin alphaVbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466505(US10799605, Example 19)
Affinity DataIC50:  12.6nMAssay Description:Ca2+ ions are usually kept at nanomolar levels in the cytosol of cells, and act in a number of signal transduction pathways as second messengers. Man...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423727(CHEMBL593226)
Affinity DataIC50:  13nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423734(CHEMBL591779)
Affinity DataIC50:  13nMAssay Description:Inhibition of integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217421((S)-3-(2-((3R,5S)-1-(methoxycarbonyl)-5-((pyridin-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217420(12S,14R,30S-4-{[2-carboxy-2-(2,4,6-trimethylbenzen...)
Affinity DataIC50:  16nMAssay Description:Inhibition of integrin alphaVbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466502(US10799605, Example 13)
Affinity DataIC50:  17.5nMAssay Description:Ca2+ ions are usually kept at nanomolar levels in the cytosol of cells, and act in a number of signal transduction pathways as second messengers. Man...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50217435(2S,4R,20S-4-{[2-carboxy-2-(2,4,6-trimethyl-benzene...)
Affinity DataIC50:  19nMAssay Description:Inhibition of integrin alphaVbeta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
3B Pharmaceuticals

US Patent
LigandPNGBDBM466500(US10799605, Example 5)
Affinity DataIC50:  20nMAssay Description:Ca2+ ions are usually kept at nanomolar levels in the cytosol of cells, and act in a number of signal transduction pathways as second messengers. Man...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423720(CHEMBL606866)
Affinity DataIC50: >20nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423732(CHEMBL590389)
Affinity DataIC50:  21nMAssay Description:Inhibition of integrin alpha5beta1 receptor-mediated HEK293 cell adhesionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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