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Found 178 with Last Name = 'otaka' and Initial = 'a'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50127171(CHEMBL299578 | N-{3-[(4-Amino-benzenesulfonyl)-iso...)
Affinity DataKi:  0.100nMAssay Description:Inhibitory activity of the compound against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM810((3S,4aS,8aS)-N-tert-butyl-2-[(2R,3S)-2-hydroxy-3-[...)
Affinity DataKi:  0.120nMAssay Description:Inhibitory activity of the compound against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM519((2S)-N-[(2S,3R)-4-[(3S,4aS,8aS)-3-(tert-butylcarba...)
Affinity DataKi:  0.190nMAssay Description:Inhibitory activity of the compound against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
Affinity DataKi:  0.280nMAssay Description:Inhibitory activity of the compound against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50127172(4-Amino-N-[3-benzyl-2-hydroxy-6-methanesulfonylami...)
Affinity DataKi:  0.380nMAssay Description:Inhibitory activity of the compound against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50159214(CHEMBL438934)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166087(CHEMBL436097 | N-{3-[(2R,5S,8S,14R)-5-(3-Guanidino...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50159213(CHEMBL370001 | N-{3-[10-(3-Guanidino-propyl)-4-(4-...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50102044(CHEMBL2373002 | Derivative of T140 peptide)
Affinity DataIC50:  8nMAssay Description:Inhibitory concentration determined on an HIV infection model mediated by CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166106(CHEMBL436283 | N-{3-[(2S,5S,8S,14R)-5-(3-Guanidino...)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166096(CHEMBL372874 | N-[(2S,5R,11S,14S,16aS)-14-(3-Guani...)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50096735(CHEMBL2372983 | Compound T140)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration determined on an HIV infection model mediated by CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166079(CHEMBL192183 | N-[(2R,5R,11S,14S,16aS)-14-(3-Guani...)
Affinity DataIC50:  10nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50102037(CHEMBL2372993 | Derivative of T140 peptide)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration determined on an HIV infection model mediated by CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166101(CHEMBL372422 | N-{3-[(2S,5S,11R)-14-(2-Amino-ethyl...)
Affinity DataIC50:  16nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50102036(CHEMBL2372985 | Derivative of T140 peptide)
Affinity DataIC50:  19nMAssay Description:Inhibitory concentration determined on an HIV infection model mediated by CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166086(CHEMBL192594 | N-{3-[(2S,5S,11R)-14-(3-Amino-propy...)
Affinity DataIC50:  19nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50102040(CHEMBL2372994 | T140)
Affinity DataIC50:  23nMAssay Description:Inhibitory concentration determined on an HIV infection model mediated by CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166093(CHEMBL193217 | N-{3-[(2S,5S,11R,14S)-14-(2-Guanidi...)
Affinity DataIC50:  24nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50102032(CHEMBL2373001 | Derivative of T140 peptide)
Affinity DataIC50:  24nMAssay Description:Inhibitory concentration determined on an HIV infection model mediated by CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50410271(CHEMBL2113071)
Affinity DataIC50:  32nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166080(CHEMBL192368 | N-{4-[(2S,5S,8S,14R)-5-(3-Guanidino...)
Affinity DataIC50:  33nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166094(CHEMBL373155 | N-{3-[(2S,5S,11R,14S)-11-(4-Hydroxy...)
Affinity DataIC50:  42nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50102035(CHEMBL2372997 | Derivative of T140 peptide)
Affinity DataIC50:  51nMAssay Description:Inhibitory concentration determined on an HIV infection model mediated by CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166108(CHEMBL364295 | N-{3-[(3R,6S,9S,14S)-6-(3-Guanidino...)
Affinity DataIC50:  54nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166088(CHEMBL191687 | N-{3-[(2S,5S,11R,14R)-11-(4-Hydroxy...)
Affinity DataIC50:  63nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166109(CHEMBL365952 | N-{3-[(2S,5S,11R,14R)-14-(4-Amino-b...)
Affinity DataIC50:  97nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166098(3-[(2R,5S,8S,14R)-5-(3-Guanidino-propyl)-14-(4-hyd...)
Affinity DataIC50:  170nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50410273(CHEMBL2113070)
Affinity DataIC50:  180nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50410270(CHEMBL2112323)
Affinity DataIC50:  190nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166105(CHEMBL192685 | N-{3-[(2S,5S,11R,14S)-11-(4-Hydroxy...)
Affinity DataIC50:  230nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166092(2-[(2R,5S,8S,14R)-5-(3-Guanidino-propyl)-14-(4-hyd...)
Affinity DataIC50:  270nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50151585(CHEMBL3774476)
Affinity DataIC50:  280nMAssay Description:Inhibition of full length N-terminal His-tagged human recombinant LSD1 (1 to 852 residues) expressed in Escherichia coli BL21(DE3) cells using H3K4me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50151584(CHEMBL3775613)
Affinity DataIC50:  290nMAssay Description:Inhibition of full length N-terminal His-tagged human recombinant LSD1 (1 to 852 residues) expressed in Escherichia coli BL21(DE3) cells using H3K4me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50151583(CHEMBL3774920)
Affinity DataIC50:  320nMAssay Description:Inhibition of full length N-terminal His-tagged human recombinant LSD1 (1 to 852 residues) expressed in Escherichia coli BL21(DE3) cells using H3K4me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166097(CHEMBL424826 | N-{3-[(5R,11S,14S,16aR)-5-(4-Hydrox...)
Affinity DataIC50:  420nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50151587(CHEMBL3774486)
Affinity DataIC50:  440nMAssay Description:Inhibition of full length N-terminal His-tagged human recombinant LSD1 (1 to 852 residues) expressed in Escherichia coli BL21(DE3) cells using H3K4me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166102(CHEMBL371993 | N-{3-[(2S,5S,11R,14R)-11-(4-Hydroxy...)
Affinity DataIC50:  490nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166091((4S,7S,10S,13R)-13-(3-Guanidino-propionylamino)-10...)
Affinity DataIC50:  530nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerpin H1(Mus musculus)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50320837(CHEMBL1163302)
Affinity DataIC50:  580nMAssay Description:Binding affinity to mouse recombinant HSP47 expressed in Escherichia coli JM109 after 10 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50151588(CHEMBL3775735)
Affinity DataIC50:  610nMAssay Description:Inhibition of full length N-terminal His-tagged human recombinant LSD1 (1 to 852 residues) expressed in Escherichia coli BL21(DE3) cells using H3K4me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166107(3-[(2R,5S,8S,14R)-5-(3-Guanidino-propyl)-14-(4-hyd...)
Affinity DataIC50:  610nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerpin H1(Mus musculus)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50320838(CHEMBL1163304)
Affinity DataIC50:  640nMAssay Description:Binding affinity to mouse recombinant HSP47 expressed in Escherichia coli JM109 after 10 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166090((R)-13-(3-Guanidino-propionylamino)-10-(3-guanidin...)
Affinity DataIC50:  690nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerpin H1(Mus musculus)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50320839(CHEMBL2372617)
Affinity DataIC50:  690nMAssay Description:Binding affinity to mouse recombinant HSP47 expressed in Escherichia coli JM109 after 10 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerpin H1(Mus musculus)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50320841(CHEMBL1163305)
Affinity DataIC50:  940nMAssay Description:Binding affinity to mouse recombinant HSP47 expressed in Escherichia coli JM109 after 10 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerpin H1(Mus musculus)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50320840(CHEMBL1163301)
Affinity DataIC50:  940nMAssay Description:Binding affinity to mouse recombinant HSP47 expressed in Escherichia coli JM109 after 10 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166099(CHEMBL362983 | N-{3-[(Z)-(3R,6S,9S,14R)-6-(3-Guani...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166081((4S,7S,10S,13R)-10-(3-Guanidino-propyl)-13-(3-guan...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166083(CHEMBL191869 | N-{3-[(3R,6R,9S,14S)-6-(3-Guanidino...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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