Affinity DataKi: 0.0140nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of endomorphin-2 binding to rat brain mu opioid reeceptorMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to mouse brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of endomorphin-2 binding to rat brain mu opioid reeceptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to mouse brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to mouse brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(GUINEA PIG)
Hungarian Academy of Sciences
Curated by PDSP Ki Database
Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy of Sciences
Curated by PDSP Ki Database
Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy of Sciences
Curated by PDSP Ki Database
Hungarian Academy of Sciences
Curated by PDSP Ki Database
Affinity DataKi: 9.5nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy of Sciences
Curated by PDSP Ki Database
Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy of Sciences
Curated by PDSP Ki Database
Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to mouse brain mu opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy of Sciences
Curated by PDSP Ki Database
Hungarian Academy of Sciences
Curated by PDSP Ki Database
Affinity DataKi: 26nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to mouse brain mu opioid receptorMore data for this Ligand-Target Pair