Affinity DataIC50: 0.110nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 8.20nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against hepatitis C virus NS5B polymerase enzyme; Range=6-9 nMMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against hepatitis C virus NS5B polymerase enzyme; Range=6-9 nMMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against hepatitis C virus NS5B polymerase enzyme; Range=6-9 nMMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against hepatitis C virus NS5B polymerase enzyme; Range=6-9 nMMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against hepatitis C virus NS5B polymerase enzyme; Range=6-9 nMMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of Trypanosoma cruzi CYP51More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Irbm (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibitory activity against by hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of Trypanosoma cruzi CYP51More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of Trypanosoma cruzi CYP51More data for this Ligand-Target Pair