Affinity DataKi: 9.10nM ΔG°: -45.4kJ/mole IC50: 34.3nMpH: 7.0 T: 2°CAssay Description:In vitro kinase inhibition assay using purified GSK-3 alpha from insect cells, was incubated at room temperature with substrate, and test compounds i...More data for this Ligand-Target Pair
Affinity DataKi: 30.8nM ΔG°: -42.4kJ/mole IC50: 77.5nMpH: 7.0 T: 2°CAssay Description:In vitro kinase inhibition assay using purified GSK-3 alpha from insect cells, was incubated at room temperature with substrate, and test compounds i...More data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Inhibitory activity was tested agianst rat ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Inhibitory activity was tested agianst rat ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 710nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibitory activity was tested agianst human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibitory activity was tested agianst rat ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Inhibitory activity was tested agianst ATP-Citrate Lyase (ACL) enzyme in ratMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Inhibition of recombinant ATP-Citrate Lyase activity as maleate dehydrogenase catalyzed reduction of oxaloacetate by NADHMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 5.70E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibition of recombinant ATP-Citrate Lyase activity as maleate dehydrogenase catalyzed reduction of oxaloacetate by NADHMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair
Affinity DataKi: 7.30E+3nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair
Affinity DataKi: 7.40E+3nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair
Affinity DataKi: 9.50E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Inhibition of recombinant ATP-Citrate Lyase activity as maleate dehydrogenase catalyzed reduction of oxaloacetate by NADHMore data for this Ligand-Target Pair
TargetCathepsin B(Homo sapiens (Human))
S£O Carlos Institute Of Chemistry-University Of S£O Paulo (Iqsc-Usp)
Curated by ChEMBL
S£O Carlos Institute Of Chemistry-University Of S£O Paulo (Iqsc-Usp)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
TargetCathepsin B(Homo sapiens (Human))
S£O Carlos Institute Of Chemistry-University Of S£O Paulo (Iqsc-Usp)
Curated by ChEMBL
S£O Carlos Institute Of Chemistry-University Of S£O Paulo (Iqsc-Usp)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
TargetCathepsin B(Homo sapiens (Human))
S£O Carlos Institute Of Chemistry-University Of S£O Paulo (Iqsc-Usp)
Curated by ChEMBL
S£O Carlos Institute Of Chemistry-University Of S£O Paulo (Iqsc-Usp)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
TargetCathepsin B(Homo sapiens (Human))
S£O Carlos Institute Of Chemistry-University Of S£O Paulo (Iqsc-Usp)
Curated by ChEMBL
S£O Carlos Institute Of Chemistry-University Of S£O Paulo (Iqsc-Usp)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair
Affinity DataKi: 1.05E+4nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Inhibitory activity was tested agianst ATP-Citrate Lyase (ACL) enzyme in ratMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Inhibitory activity against rat ATP-citrate lyase activity by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADH.More data for this Ligand-Target Pair