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Found 87 with Last Name = 'pemp' and Initial = 'd'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056333(CHEMBL3322470)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056338(CHEMBL3322475)
Affinity DataKi:  1.27E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056339(CHEMBL3322476)
Affinity DataKi:  3.10E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160434((6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-indol-3-...)
Affinity DataEC50:  603nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataEC50:  741nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048479(CHEMBL3310159)
Affinity DataEC50:  3.16E+4nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048480(CHEMBL3310161)
Affinity DataEC50:  6.61E+3nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048481(CHEMBL3310162)
Affinity DataEC50:  1.20E+4nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048482(CHEMBL3310163)
Affinity DataEC50:  5.75E+4nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048483(CHEMBL3310164)
Affinity DataEC50:  1.95E+4nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048484(CHEMBL3310166)
Affinity DataEC50:  1.66E+4nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048486(CHEMBL3310167)
Affinity DataEC50:  2.88E+3nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP by scint...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50244276(2-(4-ethoxybenzyl)-N,N-diethyl-1-isopentyl-1H-benz...)
Affinity DataEC50:  141nMAssay Description:Agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048487(CHEMBL3310157)
Affinity DataEC50:  174nMAssay Description:Agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048488(CHEMBL3310158)
Affinity DataEC50:  295nMAssay Description:Agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048489(CHEMBL3310160)
Affinity DataEC50:  1.26E+4nMAssay Description:Antagonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM21279(1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N...)
Affinity DataEC50:  58nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048479(CHEMBL3310159)
Affinity DataEC50:  2.51E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048480(CHEMBL3310161)
Affinity DataEC50:  6.31E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048481(CHEMBL3310162)
Affinity DataEC50:  3.47E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048483(CHEMBL3310164)
Affinity DataEC50:  2.40E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048484(CHEMBL3310166)
Affinity DataEC50:  2.57E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048486(CHEMBL3310167)
Affinity DataEC50:  1.74E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP by scint...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50244276(2-(4-ethoxybenzyl)-N,N-diethyl-1-isopentyl-1H-benz...)
Affinity DataEC50:  3.24E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50048487(CHEMBL3310157)
Affinity DataEC50:  1.35E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056317(CHEMBL3322349)
Affinity DataEC50:  112nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056318(CHEMBL3322350)
Affinity DataEC50:  3.85E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50328952(CHEMBL1269766 | N,N'-(Iminodiheptane-7,1-diyl)bis[...)
Affinity DataEC50:  871nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056319(CHEMBL3322458)
Affinity DataEC50:  1.35E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056320(CHEMBL3322454)
Affinity DataEC50:  1.50E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056321(CHEMBL3322455)
Affinity DataEC50:  4.07E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056322(CHEMBL3322457)
Affinity DataEC50:  9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056323(CHEMBL3322459)
Affinity DataEC50:  9.66E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056324(CHEMBL3322460)
Affinity DataEC50:  8.71E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056325(CHEMBL3322461)
Affinity DataEC50:  8.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056326(CHEMBL3322462)
Affinity DataEC50:  7.60E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056327(CHEMBL3322463)
Affinity DataEC50:  2.43E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056328(CHEMBL3322464)
Affinity DataEC50:  3.16E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056329(CHEMBL3322465)
Affinity DataEC50:  1.05E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056330(CHEMBL3322467)
Affinity DataEC50:  1.62E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056331(CHEMBL3322468)
Affinity DataEC50:  7.24E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056332(CHEMBL3322469)
Affinity DataEC50:  8.85E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056333(CHEMBL3322470)
Affinity DataEC50:  2.95E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056334(CHEMBL3322471)
Affinity DataEC50:  776nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056335(CHEMBL3322472)
Affinity DataEC50:  501nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056336(CHEMBL3322473)
Affinity DataEC50:  110nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056337(CHEMBL3322474)
Affinity DataEC50:  1.10E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056338(CHEMBL3322475)
Affinity DataEC50:  661nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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