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Found 38 with Last Name = 'pendley' and Initial = 'ce'
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000485((S)-2-(5-chlorospiro[2,3-dihydrobenzo[b]furan-2,1'...)
Affinity DataKi:  0.190nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82403(CAS_108186 | CI-988 | NSC_108186)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82404(Glycinamide,N-[[[3-(2-sulfoethyl)phenyl]amino]carb...)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82404(Glycinamide,N-[[[3-(2-sulfoethyl)phenyl]amino]carb...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000482((R)-2-(5-chlorospiro[2,3-dihydrobenzo[b]furan-2,1'...)
Affinity DataKi:  0.890nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000480(2-(5-chlorospiro[2,3-dihydrobenzo[b]furan-2,1'-cyc...)
Affinity DataKi:  1.10nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000479(7-Chloro-2,3,4,5-tetrahydro-benzo[b]oxepine-9-carb...)
Affinity DataKi:  1.20nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000492((zacopride)4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataKi:  1.5nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000495((ICS 205-930)1H-Indole-3-carboxylic acid 6-methyl-...)
Affinity DataKi:  1.70nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000483((BRL 43694)1-Methyl-1H-indazole-3-carboxylic acid ...)
Affinity DataKi:  1.70nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82403(CAS_108186 | CI-988 | NSC_108186)
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000494(7-Bromo-2,3,4,5-tetrahydro-benzo[b]oxepine-9-carbo...)
Affinity DataKi:  2.20nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82241(CAS_5534-95-2 | NSC_444007 | Pentagastrin)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000487(8-Chloro-3,4,5,6-tetrahydro-2H-benzo[b]oxocine-10-...)
Affinity DataKi:  4.70nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM50061220(1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  4.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82241(CAS_5534-95-2 | NSC_444007 | Pentagastrin)
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000489(CHEMBL353993 | N-(1-Aza-bicyclo[2.2.2]oct-3-yl)-5-...)
Affinity DataKi:  6.10nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  6.20nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM50061220(1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  7.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000478(2,3,4,5-Tetrahydro-benzo[b]oxepine-9-carboxylic ac...)
Affinity DataKi:  14nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000484(7-Chloro-2,2-dimethyl-2,3,4,5-tetrahydro-benzo[b]o...)
Affinity DataKi:  16nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000486(CHEMBL368992 | N-(1-Aza-bicyclo[2.2.2]oct-3-yl)-2-...)
Affinity DataKi: >30nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000488(CHEMBL171070 | N-(1-Aza-bicyclo[2.2.2]oct-3-yl)-5-...)
Affinity DataKi:  47nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000490(7-Chloro-2,3,4,5-tetrahydro-benzo[b]oxepine-9-carb...)
Affinity DataKi:  63nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  87nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50000481(8-Amino-7-chloro-2,3,4,5-tetrahydro-benzo[b]oxepin...)
Affinity DataKi: >100nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  141nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))
Affinity DataKi:  883nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM48320(4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-metho...)
Affinity DataKi:  995nMAssay Description:Displacement of the 5-hydroxytryptamine 3 receptor ligand [3H]GR-65630 from rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82403(CAS_108186 | CI-988 | NSC_108186)
Affinity DataKi:  1.44E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM82404(Glycinamide,N-[[[3-(2-sulfoethyl)phenyl]amino]carb...)
Affinity DataKi:  1.63E+3nMMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM50008673(2-(4-Chloro-benzoylamino)-3-(1H-indol-3-yl)-propio...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholecystokinin(GUINEA PIG)
Rhone-Poulenc Rorer Central Research

Curated by PDSP Ki Database
LigandPNGBDBM50008673(2-(4-Chloro-benzoylamino)-3-(1H-indol-3-yl)-propio...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed