TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot
Curated by ChEMBL
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Displacement of [3H]rosiglitazone from N-terminal His-tagged human PPARgamma ligand binding domain expressed in Escherichia coli BL21 DE3 cells by sc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot
Curated by ChEMBL
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot
Curated by ChEMBL
Affinity DataKi: 88nMAssay Description:Displacement of [3H]rosiglitazone from N-terminal His-tagged human PPARgamma ligand binding domain expressed in Escherichia coli BL21 DE3 cells by sc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot
Curated by ChEMBL
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot
Curated by ChEMBL
Affinity DataKi: 971nMAssay Description:Displacement of [3H]rosiglitazone from N-terminal His-tagged human PPARgamma ligand binding domain expressed in Escherichia coli BL21 DE3 cells by sc...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FAAH in Wistar rat brain intact neurons assessed as reduction in [3H]anandamide hydrolysis using [3H]anandamide as substrate preincubat...More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of FAAH in Wistar rat brain membranes assessed as reduction in [3H]anandamide hydrolysis using [3H]anandamide as substrate preincubated fo...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bari Aldo Moro
Curated by ChEMBL
University Of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated with enzyme for 10 mins followed by substrate addition for 2 hrs by fluor...More data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bari Aldo Moro
Curated by ChEMBL
University Of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of recombinant human C-terminal FLAG-tagged FAAH expressed in HEK293T cells preincubated for 4 hrs followed by addition of FP-TAMRA probe ...More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 103nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 122nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 135nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 136nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 189nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 503nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 509nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 595nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 735nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 767nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 969nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 993nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant human MMP13 catalytic domain (Tyr104 to Asn274 residues) expressed in Escherichia coli cells using Mca-Pro-Leu-Gly-Leu-Dpa-...More data for this Ligand-Target Pair
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human MMP13 catalytic domain (Tyr104 to Asn274 residues) expressed in Escherichia coli cells using Mca-Pro-Leu-Gly-Leu-Dpa-...More data for this Ligand-Target Pair
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) expressed in yeast cells using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2/...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) expressed in yeast cells using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2/...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) expressed in yeast cells using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2/...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of recombinant human MMP13 catalytic domain (Tyr104 to Asn274 residues) expressed in Escherichia coli cells using Mca-Pro-Leu-Gly-Leu-Dpa-...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of recombinant human MMP13 catalytic domain (Tyr104 to Asn274 residues) expressed in Escherichia coli cells using Mca-Pro-Leu-Gly-Leu-Dpa-...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) expressed in yeast cells using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2/...More data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.08E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.58E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bari Aldo Moro
Curated by ChEMBL
University Of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of FAAH (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.61E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair