Compile Data Set for Download or QSAR
maximum 50k data
Found 607 with Last Name = 'piemontese' and Initial = 'l'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]rosiglitazone from N-terminal His-tagged human PPARgamma ligand binding domain expressed in Escherichia coli BL21 DE3 cells by sc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot

Curated by ChEMBL
LigandPNGBDBM28762((2R)-2-(4-{2-[1,3-benzoxazol-2-yl(heptyl)amino]eth...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]rosiglitazone from N-terminal His-tagged human PPARgamma ligand binding domain expressed in Escherichia coli BL21 DE3 cells by sc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot

Curated by ChEMBL
LigandPNGBDBM28763((2S)-2-(4-{2-[1,3-benzoxazol-2-yl(heptyl)amino]eth...)
Affinity DataKi:  971nMAssay Description:Displacement of [3H]rosiglitazone from N-terminal His-tagged human PPARgamma ligand binding domain expressed in Escherichia coli BL21 DE3 cells by sc...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM26739(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of FAAH in Wistar rat brain intact neurons assessed as reduction in [3H]anandamide hydrolysis using [3H]anandamide as substrate preincubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593777(CHEMBL5185868)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593778(CHEMBL5189408)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM26739(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of FAAH in Wistar rat brain membranes assessed as reduction in [3H]anandamide hydrolysis using [3H]anandamide as substrate preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50307083(4-nitrophenyl 4-(3-phenoxybenzyl)piperazine-1-carb...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated with enzyme for 10 mins followed by substrate addition for 2 hrs by fluor...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593779(CHEMBL5193520)
Affinity DataIC50:  42nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50505364(CHEMBL4460898)
Affinity DataIC50:  49nMAssay Description:Inhibition of recombinant human C-terminal FLAG-tagged FAAH expressed in HEK293T cells preincubated for 4 hrs followed by addition of FP-TAMRA probe ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593781(CHEMBL5190969)
Affinity DataIC50:  90nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593768(CHEMBL5195980)
Affinity DataIC50:  103nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593767(CHEMBL5207120)
Affinity DataIC50:  122nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593773(CHEMBL5182803)
Affinity DataIC50:  135nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593780(CHEMBL5209013)
Affinity DataIC50:  136nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593785(CHEMBL5169781)
Affinity DataIC50:  189nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593784(CHEMBL5175715)
Affinity DataIC50:  300nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593780(CHEMBL5209013)
Affinity DataIC50:  503nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593769(CHEMBL5180014)
Affinity DataIC50:  509nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593771(CHEMBL5178350)
Affinity DataIC50:  595nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593776(CHEMBL5204532)
Affinity DataIC50:  735nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593770(CHEMBL5202267)
Affinity DataIC50:  767nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593774(CHEMBL5177371)
Affinity DataIC50:  880nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593783(CHEMBL5185234)
Affinity DataIC50:  900nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593776(CHEMBL5204532)
Affinity DataIC50:  969nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593782(CHEMBL5206245)
Affinity DataIC50:  993nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593770(CHEMBL5202267)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593772(CHEMBL5203325)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593777(CHEMBL5185868)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593775(CHEMBL5175950)
Affinity DataIC50:  1.68E+3nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593766(CHEMBL5170984)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCollagenase 3(Homo sapiens (Human))
"A. Moro" University Of Bari

Curated by ChEMBL
LigandPNGBDBM50541090(CHEMBL4647123)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of recombinant human MMP13 catalytic domain (Tyr104 to Asn274 residues) expressed in Escherichia coli cells using Mca-Pro-Leu-Gly-Leu-Dpa-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593785(CHEMBL5169781)
Affinity DataIC50:  2.15E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCollagenase 3(Homo sapiens (Human))
"A. Moro" University Of Bari

Curated by ChEMBL
LigandPNGBDBM50541091(CHEMBL4639311)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of recombinant human MMP13 catalytic domain (Tyr104 to Asn274 residues) expressed in Escherichia coli cells using Mca-Pro-Leu-Gly-Leu-Dpa-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593771(CHEMBL5178350)
Affinity DataIC50:  2.22E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
"A. Moro" University Of Bari

Curated by ChEMBL
LigandPNGBDBM50541092(CHEMBL4634914)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) expressed in yeast cells using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
"A. Moro" University Of Bari

Curated by ChEMBL
LigandPNGBDBM50541090(CHEMBL4647123)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) expressed in yeast cells using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
"A. Moro" University Of Bari

Curated by ChEMBL
LigandPNGBDBM50541091(CHEMBL4639311)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) expressed in yeast cells using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
"A. Moro" University Of Bari

Curated by ChEMBL
LigandPNGBDBM50541093(CHEMBL4640667)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of recombinant human MMP13 catalytic domain (Tyr104 to Asn274 residues) expressed in Escherichia coli cells using Mca-Pro-Leu-Gly-Leu-Dpa-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
"A. Moro" University Of Bari

Curated by ChEMBL
LigandPNGBDBM50541092(CHEMBL4634914)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of recombinant human MMP13 catalytic domain (Tyr104 to Asn274 residues) expressed in Escherichia coli cells using Mca-Pro-Leu-Gly-Leu-Dpa-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593781(CHEMBL5190969)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
"A. Moro" University Of Bari

Curated by ChEMBL
LigandPNGBDBM50541104(CHEMBL1483847)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) expressed in yeast cells using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2/...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593767(CHEMBL5207120)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593778(CHEMBL5189408)
Affinity DataIC50:  5.01E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593773(CHEMBL5182803)
Affinity DataIC50:  5.08E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593766(CHEMBL5170984)
Affinity DataIC50:  5.58E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM22987((5Z,8Z,11Z,14Z)-N-[2-(5-hydroxy-1H-indol-3-yl)ethy...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of FAAH (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50593775(CHEMBL5175950)
Affinity DataIC50:  5.61E+3nMAssay Description:Inhibition of human BuChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Displayed 1 to 50 (of 607 total ) | Next | Last >>
Jump to: