TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 640nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 850nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 910nMAssay Description:Competitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 970nMAssay Description:Competitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.26E+3nM IC50: 1.67E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.28E+3nM IC50: 1.39E+3nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.54E+3nM IC50: 1.36E+3nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.67E+3nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3.77E+3nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3.77E+3nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3.84E+3nMAssay Description:Competitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3.99E+3nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 4.10E+3nM IC50: 490nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 5.06E+3nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 5.45E+3nM IC50: 4.36E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 5.67E+3nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 5.68E+3nMAssay Description:Competitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 7.60E+3nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 8.36E+3nMAssay Description:Uncompetitive inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured up to 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 8.95E+3nM IC50: 5.11E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 9.04E+3nM IC50: 2.75E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 9.90E+3nM IC50: 1.03E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.58E+4nM IC50: 5.73E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.95E+4nM IC50: 1.07E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3.48E+4nM IC50: 1.56E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 4.37E+4nM IC50: 1.66E+3nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 4.68E+4nM IC50: 3.02E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.17E+5nM IC50: 7.98E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.31E+5nM IC50: 5.34E+3nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 20 mins prior to substrate addition by Ellmans met...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of acetylcholinesterase (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of acetylcholinesterase in Albino LACA mouse brain homogenates using acetylthiocholine iodide as substrate measured for 2 mins by Ellman's...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.42E+3nMAssay Description:Inhibition of acetylcholinesterase in Albino LACA mouse brain homogenates using acetylthiocholine iodide as substrate measured for 2 mins by Ellman's...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.03E+3nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 4.09E+3nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of acetylcholinesterase in Albino LACA mouse brain homogenates using acetylthiocholine iodide as substrate measured for 2 mins by Ellman's...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 7.09E+3nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of acetylcholinesterase in Albino LACA mouse brain homogenates using acetylthiocholine iodide as substrate measured for 2 mins by Ellman's...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of acetylcholinesterase in Albino LACA mouse brain homogenates using acetylthiocholine iodide as substrate measured for 2 mins by Ellman's...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of albino mouse brain AChE using acetylthiocholine iodide as substrate measured for 2 mins by Ellmans methodMore data for this Ligand-Target Pair