Affinity DataKi: 0.0290nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-1A adrenergic receptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0580nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-1D adrenergic receptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-1A adrenergic receptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-1B adrenergic receptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.850nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-1D adrenergic receptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-1D adrenergic receptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-1A adrenergic receptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.68nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-1B adrenergic receptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity against rat Alpha-2B adrenergic receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.95nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-1B adrenergic receptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinity against rat Alpha-2B adrenergic receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity against human Alpha-2C adrenergic receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 13.1nMAssay Description:Binding affinity against rat Alpha-2B adrenergic receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 13.4nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-2A adrenergic receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 16.6nMAssay Description:Binding affinity against human Alpha-2C adrenergic receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 19.7nMAssay Description:Binding affinity against Dopamine receptor D2 using [3H]-spiroperidol as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity against human Alpha-2C adrenergic receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 94.9nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-2A adrenergic receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 717nMAssay Description:Binding affinity against Dopamine receptor D1 using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity against human adrenergic receptor subtype Alpha-2A adrenergic receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.38E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 1 receptor using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.87E+3nMAssay Description:Binding affinity against adrenergic receptor subtype Beta-2 adrenergic receptor using [3H]-DHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.06E+4nMAssay Description:Binding affinity against Beta-1 adrenergic receptor using [3H]-DHA as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of mouse DGAT1 using [1-14C]decanoyl-CoA substrate by phospholipid flash plate assayMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of human DGAT1 expressed in human HeLa cells assessed as reduction in triglyceride synthesisMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant DGAT2 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid flash plate assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant DGAT1 expressed in insect cell membrane using [1-14C]decanoyl-CoA substrate by phospholipid fl...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human ERG by manual patch clamp assayMore data for this Ligand-Target Pair