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Found 221 with Last Name = 'pomper' and Initial = 'm'
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by radiometric assayMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by fluorescence-based assayMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456924(US10736974, Compound YC-I-27)
Affinity DataKi:  0.0100nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456928(US10736974, Compound XY-44)
Affinity DataKi:  0.0170nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456930(US10736974, Compound XY-59)
Affinity DataKi:  0.0200nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456923(US10736974, Compound DCIBC)
Affinity DataKi:  0.0300nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578399(US11478558, Compound L9)
Affinity DataKi:  0.0350nMAssay Description:TBDMore data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456931(US10736974, Compound XY-58)
Affinity DataKi:  0.0360nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456929(US10736974, Compound XY-45)
Affinity DataKi:  0.100nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578398(US11478558, Compound L8)
Affinity DataKi:  0.120nMAssay Description:TBDMore data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50246934((S)-2-(3-((S)-1-carboxy-5-(4-fluorobenzamido)penty...)
Affinity DataKi:  0.194nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298756((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50246934((S)-2-(3-((S)-1-carboxy-5-(4-fluorobenzamido)penty...)
Affinity DataKi:  0.256nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456920(US10736974, Entry 23)
Affinity DataKi:  0.260nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578392(US11478558, Compound L2)
Affinity DataKi:  0.265nMAssay Description:TBDMore data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578394(US11478558, Compound L4)
Affinity DataKi:  0.265nMAssay Description:TBDMore data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456925(US10736974, Compound YC-I-26)
Affinity DataKi:  0.300nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456914(US10736974, Compound XY-43 | US10736974, Entry 17)
Affinity DataKi:  0.320nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456914(US10736974, Compound XY-43 | US10736974, Entry 17)
Affinity DataKi:  0.320nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456927(US10736974, Compound C8)
Affinity DataKi:  0.350nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50246935((S)-2-(3-((S)-1-carboxy-5-(3-iodonicotinamido)pent...)
Affinity DataKi:  0.351nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456921(US10736974, Entry 24)
Affinity DataKi:  0.400nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578391(US11478558, Compound 3)
Affinity DataKi:  0.430nMAssay Description:TBDMore data for this Ligand-Target Pair
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In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578395(US11478558, Compound L5)
Affinity DataKi:  0.545nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578397(US11478558, Compound L7)
Affinity DataKi:  0.550nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50246935((S)-2-(3-((S)-1-carboxy-5-(3-iodonicotinamido)pent...)
Affinity DataKi:  0.557nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578396(US11478558, Compound L6)
Affinity DataKi:  0.640nMAssay Description:TBDMore data for this Ligand-Target Pair
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50304738(2-(3-((S)-1-carboxy-3-methylbutyl)ureido)pentanedi...)
Affinity DataKi:  0.75nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578400(US11478558, Compound L10)
Affinity DataKi:  0.815nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456906(US10736974, Compound XY-26 | US10736974, Entry 9)
Affinity DataKi:  0.900nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456906(US10736974, Compound XY-26 | US10736974, Entry 9)
Affinity DataKi:  0.900nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50304738(2-(3-((S)-1-carboxy-3-methylbutyl)ureido)pentanedi...)
Affinity DataKi:  1.08nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCAP cells assessed as glutamate formation using NAAG as substrate after 60 mins by fluorometric...More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456926(US10736974, Compound DCFPyL)
Affinity DataKi:  1.10nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578389(US11478558, Compound 1)
Affinity DataKi:  1.15nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578390(US11478558, Compound 2)
Affinity DataKi:  1.28nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578401(US11478558, Compound L12)
Affinity DataKi:  2.12nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298754((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298760(CHEMBL574766 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298738(CHEMBL583783 | benzyl(2S,5S,8S,11S,14S)-8-(3-amino...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM578402(US11478558, Compound L13)
Affinity DataKi:  4.17nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298761(CHEMBL574788 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  4.40nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456908(US10736974, Compound XY-28 | US10736974, Entry 11)
Affinity DataKi:  4.80nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456908(US10736974, Compound XY-28 | US10736974, Entry 11)
Affinity DataKi:  4.80nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50304722((S)-2-(3-((S)-1-Carboxybut-3-ynyl)ureido)-6-(4-iod...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50304731((S)-2-(3-((S)-1-Carboxy-2-(furan-2-yl)ethyl)ureido...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298757((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456900(US10736974, Entry 7)
Affinity DataKi:  6nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298762(CHEMBL574924 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298739(CHEMBL583784 | benzyl(2S,5S,8S,11S,14S)-14-formyl-...)
Affinity DataKi:  7.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM456911(US10736974, Entry 14)
Affinity DataKi:  8.30nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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