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Found 38 with Last Name = 'prota' and Initial = 'g'
TargetEstrogen receptor beta(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50255198((E)-3-Chloro-4-(3-fluoro-4-hydroxyphenyl)salicylal...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]estradiol from full-length human estrogen receptor beta by radiometric assay relative to estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]estradiol from purified full length human ERbeta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217078(2-hydroxy-6-methoxy-3',5'-dimethyl-biphenyl-4-carb...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]estradiol from purified full length human ERalpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217074(2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217078(2-hydroxy-6-methoxy-3',5'-dimethyl-biphenyl-4-carb...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217074(2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217077(2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217077(2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217080(2,6-dihydroxy-biphenyl-4-carboxylic acid pentyl es...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217071(2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217079(2-hydroxy-6-methoxy-3',5'-dimethyl-biphenyl-4-carb...)
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217072(2-hydroxy-6-methoxy-3',5'-dimethyl-biphenyl-4-carb...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217079(2-hydroxy-6-methoxy-3',5'-dimethyl-biphenyl-4-carb...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217076(2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217073(2,6-dimethoxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217080(2,6-dihydroxy-biphenyl-4-carboxylic acid pentyl es...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217075(2,6-dimethoxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217071(2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217072(2-hydroxy-6-methoxy-3',5'-dimethyl-biphenyl-4-carb...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217073(2,6-dimethoxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217075(2,6-dimethoxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50217076(2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at full length human ERbeta receptor expressed in human HEC-1 cells assessed as (ERE)2-pS2-luc reporter gene transcriptional activit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50255366((E)-5-(4-Hydroxyphenyl)salicylaldoxime | CHEMBL480...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at full-length human estrogen receptor alpha expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at full-length human estrogen receptor alpha expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at full-length human estrogen receptor alpha expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at full-length human estrogen receptor beta expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by luc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at full-length human estrogen receptor alpha expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by lu...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50255366((E)-5-(4-Hydroxyphenyl)salicylaldoxime | CHEMBL480...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at full-length human estrogen receptor alpha expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at full-length human estrogen receptor beta expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by luc...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50255366((E)-5-(4-Hydroxyphenyl)salicylaldoxime | CHEMBL480...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at full-length human estrogen receptor beta expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by luc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50255198((E)-3-Chloro-4-(3-fluoro-4-hydroxyphenyl)salicylal...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at full-length human estrogen receptor alpha expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50255198((E)-3-Chloro-4-(3-fluoro-4-hydroxyphenyl)salicylal...)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at full-length human estrogen receptor beta expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by luc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKd:  0.5nMAssay Description:Displacement of [3H]estradiol from human ERbetaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at full length human ERalpha receptor expressed in human HEC-1 cells assessed as (ERE)2-pS2-luc reporter gene transcriptional activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKd:  0.200nMAssay Description:Displacement of [3H]estradiol from human ERalphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50192460(4-(4-hydroxyphenyl)-N-methyl-3-phenylanthranylaldo...)
Affinity DataKd:  3.70nMAssay Description:Displacement of [3H]estradiol from human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed