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Found 100 with Last Name = 'protais' and Initial = 'p'
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50202337((S)-3-iodo-1,10-dimethoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292548((+)-(1R,1'S)-thaligrisine hydrochloride | CHEMBL45...)
Affinity DataIC50:  27nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50202340((S)-3-bromo-1,10-dimethoxy-6-methyl-5,6,6a,7-tetra...)
Affinity DataIC50:  66nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50269193(3-Chloroboldine | CHEMBL524439)
Affinity DataIC50:  81nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202337((S)-3-iodo-1,10-dimethoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50:  96nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50241488((+)-Coclaurine | (1R)-1-(4-hydroxybenzyl)-6-methox...)
Affinity DataIC50:  130nMAssay Description:Displacement of [3H]raclopride from rat striatal dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataIC50:  200nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50005548((+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50:  200nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50209211(3,8-dibromoboldine | CHEMBL388564)
Affinity DataIC50:  206nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50241488((+)-Coclaurine | (1R)-1-(4-hydroxybenzyl)-6-methox...)
Affinity DataIC50:  240nMAssay Description:Displacement of [3H]SCH-23390 from rat striatal dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292549((+)-(1R,1'S)-berbamunine hydrochloride | CHEMBL503...)
Affinity DataIC50:  300nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50202318((+)-boldine | (S)-(+)-Boldine | (S)-1,10-dimethoxy...)
Affinity DataIC50:  400nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202318((+)-boldine | (S)-(+)-Boldine | (S)-1,10-dimethoxy...)
Affinity DataIC50:  520nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM85444(CHEMBL506025 | Isotetrandrine (R,S) | Pheanthine (...)
Affinity DataIC50:  670nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50269193(3-Chloroboldine | CHEMBL524439)
Affinity DataIC50:  720nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202322((-)-anonaine | (R)-6,7,7a,8-tetrahydro-5H-benzo[g]...)
Affinity DataIC50:  800nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292474(7-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-ylam...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50292549((+)-(1R,1'S)-berbamunine hydrochloride | CHEMBL503...)
Affinity DataIC50:  1.04E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202340((S)-3-bromo-1,10-dimethoxy-6-methyl-5,6,6a,7-tetra...)
Affinity DataIC50:  1.05E+3nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292466(CHEMBL450147 | CHEMBL507970 | Dimethylgrisabine)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202300((R)-4-methoxy-6,7,7a,8-tetrahydro-5H-benzo[g][1,3]...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292466(CHEMBL450147 | CHEMBL507970 | Dimethylgrisabine)
Affinity DataIC50:  1.45E+3nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50209211(3,8-dibromoboldine | CHEMBL388564)
Affinity DataIC50:  1.91E+3nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292445(CHEMBL508011 | Isopiline)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292556((S,S)-oxandrine hydrochloride | CHEMBL445011)
Affinity DataIC50:  2.76E+3nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292467(Antioquine | Antioquine (S,R) | CHEMBL446564 | CHE...)
Affinity DataIC50:  3.18E+3nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292467(Antioquine | Antioquine (S,R) | CHEMBL446564 | CHE...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50099789(5-Benzyl-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]iso...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of [3H]-dopamine uptake in rat striatal synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50241642((+)-Obaberine | CHEMBL451211 | CHEMBL464525 | Obab...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50099789(5-Benzyl-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]iso...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of [3H]-Raclopride binding to the rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292468(CHEMBL504757 | Isotetrandrine)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50022723((+)-(S)-amphetamine | (+)-alpha-methylphenethylami...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50259928((R)-(+)-1-(4'-methoxybenzyl)-6-hydroxy-7-methoxy-1...)
Affinity DataIC50:  5.00E+3nMAssay Description:Displacement of [3H]raclopride from rat striatal dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50292548((+)-(1R,1'S)-thaligrisine hydrochloride | CHEMBL45...)
Affinity DataIC50:  5.60E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50292466(CHEMBL450147 | CHEMBL507970 | Dimethylgrisabine)
Affinity DataIC50:  5.64E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292469(CHEMBL443081 | CHEMBL501861 | O-methyldauricine)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50099787(5-Benzyl-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]iso...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of [3H]-dopamine uptake in rat striatal synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202287((R)-6,7,7a,8-tetrahydro-5H-benzo[g][1,3]dioxolo[4'...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292473(CHEMBL450155 | CHEMBL506299 | Secantioquine)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50241641((+)-Homoaromoline | CHEMBL509855 | Homoaromoline |...)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50292556((S,S)-oxandrine hydrochloride | CHEMBL445011)
Affinity DataIC50:  1.11E+4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292454(CHEMBL508081 | secocularidine)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292463((1S)-1-(4-hydroxybenzyl)-6-methoxy-1,2,3,4-tetrahy...)
Affinity DataIC50:  1.41E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50099786(1-Benzyl-2-propyl-1,2,3,4-tetrahydro-isoquinoline-...)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of [3H]-Raclopride binding to the rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50292553((R,S)-homoaromaline hydrochloride | CHEMBL443953)
Affinity DataIC50:  1.54E+4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292557((S,R)-pseudoxandrine hydrochloride | CHEMBL504303)
Affinity DataIC50:  1.62E+4nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292446((S)-1,10-Dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[...)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50099786(1-Benzyl-2-propyl-1,2,3,4-tetrahydro-isoquinoline-...)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to the rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292470(CHEMBL447018 | Dimethylpseudoxandrine)
Affinity DataIC50:  2.01E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50099788(5-Benzyl-6-propyl-5,6,7,8-tetrahydro-[1,3]dioxolo[...)
Affinity DataIC50:  2.03E+4nMAssay Description:Inhibition of [3H]-dopamine uptake in rat striatal synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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