TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane-A synthase(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane-A synthase(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]-RTX from human TRPV1 transfected in HEK293 cells after 60 mins by scintillation spectroscopic analysisMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataKi: 29nMAssay Description:Inhibition of rat ap2 by fluorescent 1,8-anilino-8-naphthalene sulfonate assayMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of rat ap2 by fluorescent 1,8-anilino-8-naphthalene sulfonate assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibition of human carbonic anhydrase 2 by ThermoFluor methodMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.100nMAssay Description:Inhibition of full length human recombinant HDAC6 incubated for 30 to 60 mins by HDAC-Glo I/II assayMore data for this Ligand-Target Pair
TargetTransient receptor potential M8 protein(Canis lupus familiaris (Dog))
Janssen Pharmaceutica
US Patent
Janssen Pharmaceutica
US Patent
Affinity DataIC50: 0.183nMAssay Description:For patch clamp experiments, HEK293 cells are stably transfected with canine TRPM8 and cultured in DMEM supplemented with 10% fetal bovine serum, 100...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human recombinant hormone sensitive lipase (HSL)More data for this Ligand-Target Pair
TargetTransient receptor potential M8 protein(Canis lupus familiaris (Dog))
Janssen Pharmaceutica
US Patent
Janssen Pharmaceutica
US Patent
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at canine TRPM8 expressed in HEK293 cells assessed as inhibition of intracellular calcium accumulation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:Inhibition of JAK2 (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
TargetTestis-specific serine/threonine-protein kinase 1(Mus musculus)
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataIC50: 0.330nMAssay Description:Inhibition of mouse TSSK1 by luminescent ADP-Glo assay kitMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant full length HDAC6 (unknown origin) using fluorophore conjugated substrate by microplate reader assayMore data for this Ligand-Target Pair
TargetTransient receptor potential M8 protein(Canis lupus familiaris (Dog))
Janssen Pharmaceutica
US Patent
Janssen Pharmaceutica
US Patent
Affinity DataIC50: 0.400nMT: 2°CAssay Description:The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Janssen Pharmaceutica
Curated by ChEMBL
Janssen Pharmaceutica
Curated by ChEMBL
Affinity DataIC50: 0.413nMAssay Description:Inhibition of human TRPM8 expressed in HEK293 cells assessed as inhibition of cold-induced channel current by whole cell electrophysiologyMore data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.460nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.510nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.530nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.540nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
TargetTransient receptor potential M8 protein(Canis lupus familiaris (Dog))
Janssen Pharmaceutica
US Patent
Janssen Pharmaceutica
US Patent
Affinity DataIC50: 0.554nMAssay Description:For patch clamp experiments, HEK293 cells are stably transfected with canine TRPM8 and cultured in DMEM supplemented with 10% fetal bovine serum, 100...More data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.560nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.580nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetTransient receptor potential M8 protein(Canis lupus familiaris (Dog))
Janssen Pharmaceutica
US Patent
Janssen Pharmaceutica
US Patent
Affinity DataIC50: 0.600nMT: 2°CAssay Description:The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi...More data for this Ligand-Target Pair
TargetTransient receptor potential M8 protein(Canis lupus familiaris (Dog))
Janssen Pharmaceutica
US Patent
Janssen Pharmaceutica
US Patent
Affinity DataIC50: 0.600nMT: 2°CAssay Description:The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi...More data for this Ligand-Target Pair
TargetTransient receptor potential M8 protein(Canis lupus familiaris (Dog))
Janssen Pharmaceutica
US Patent
Janssen Pharmaceutica
US Patent
Affinity DataIC50: 0.600nMAssay Description:Antagonist activity at canine TRPM8 expressed in HEK293 cells assessed as inhibition of intracellular calcium accumulation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.650nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.650nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 0.660nMAssay Description:Inhibition of wild type EGFR (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair