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Found 93 with Last Name = 'radwan' and Initial = 'mm'
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50067734((-)-(6aR-trans)-6,6,9-trimethyl-3-pentyl-6a,7,10,1...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092347(CHEMBL3586106)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092347(CHEMBL3586106)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092343(CHEMBL3586110)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM84880(THC, 8 beta-OH)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50067734((-)-(6aR-trans)-6,6,9-trimethyl-3-pentyl-6a,7,10,1...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM84880(THC, 8 beta-OH)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092345(CHEMBL3586108)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092345(CHEMBL3586108)
Affinity DataKi:  129nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092344(CHEMBL3586109)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092344(CHEMBL3586109)
Affinity DataKi:  335nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092346(CHEMBL3586107)
Affinity DataKi:  830nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092343(CHEMBL3586110)
Affinity DataKi:  912nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092348(CHEMBL3586104)
Affinity DataKi:  1.91E+3nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092342(CHEMBL3586111)
Affinity DataKi:  2.14E+3nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092348(CHEMBL3586104)
Affinity DataKi:  3.22E+3nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092346(CHEMBL3586107)
Affinity DataKi:  3.27E+3nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50092342(CHEMBL3586111)
Affinity DataKi:  5.67E+3nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50491190(CHEMBL2375656)
Affinity DataKi:  7.31E+3nMAssay Description:Displacement of [3H]-enkephalin from human delta opioid receptor transfected in CHOK1 cells after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataIC50:  292nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataIC50:  298nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269543(CHEMBL4068985)
Affinity DataIC50:  350nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211660(CHEMBL3915254)
Affinity DataIC50:  350nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269553(CHEMBL4104828)
Affinity DataIC50:  353nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211669(CHEMBL3943220)
Affinity DataIC50:  369nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269548(CHEMBL4069917)
Affinity DataIC50:  369nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269511(CHEMBL4072706)
Affinity DataIC50:  371nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269510(CHEMBL4085687)
Affinity DataIC50:  402nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269552(CHEMBL4080597)
Affinity DataIC50:  408nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269542(CHEMBL4093428)
Affinity DataIC50:  434nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50549123(CHEMBL4779272)
Affinity DataIC50:  452nMAssay Description:Inhibition of human VEGFR2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269549(CHEMBL4097121)
Affinity DataIC50:  464nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211676(CHEMBL3899514)
Affinity DataIC50:  482nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211656(CHEMBL3959627)
Affinity DataIC50:  491nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269551(CHEMBL4088467)
Affinity DataIC50:  590nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50468489(CHEMBL1305588)
Affinity DataIC50:  680nMAssay Description:Inhibition of human topoisomerase 2 using supercoiled pHOT1 DNA as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50549119(CHEMBL4763393)
Affinity DataIC50:  684nMAssay Description:Inhibition of human VEGFR2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50549115(CHEMBL4784161)
Affinity DataIC50:  707nMAssay Description:Inhibition of human VEGFR2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50549116(CHEMBL4781567)
Affinity DataIC50:  721nMAssay Description:Inhibition of human VEGFR2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50468484(CHEMBL4288104)
Affinity DataIC50:  850nMAssay Description:Inhibition of human topoisomerase 2 using supercoiled pHOT1 DNA as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM22984((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...)
Affinity DataIC50:  880nMAssay Description:Inhibition of human topoisomerase 2 using supercoiled pHOT1 DNA as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50468485(CHEMBL4286850)
Affinity DataIC50:  940nMAssay Description:Inhibition of human topoisomerase 2 using supercoiled pHOT1 DNA as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50269550(CHEMBL4089408)
Affinity DataIC50:  980nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50549122(CHEMBL4794044)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human VEGFR2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50549124(CHEMBL4777885)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of human VEGFR2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50468490(CHEMBL4291398)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of human topoisomerase 2 using supercoiled pHOT1 DNA as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50549117(CHEMBL4749461)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of human VEGFR2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211677(CHEMBL3977442)
Affinity DataIC50:  1.14E+3nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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