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Found 54 with Last Name = 'rajak' and Initial = 'h'
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354789(CHEMBL1834469)
Affinity DataIC50:  6nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354781(CHEMBL1834462)
Affinity DataIC50:  6nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354800(CHEMBL1834480)
Affinity DataIC50:  7nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354797(CHEMBL1834477)
Affinity DataIC50:  7nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354799(CHEMBL1834479)
Affinity DataIC50:  8nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354792(CHEMBL1834472)
Affinity DataIC50:  8nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354788(CHEMBL1834468)
Affinity DataIC50:  8nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354782(CHEMBL1834461)
Affinity DataIC50:  9nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354786(CHEMBL1834466)
Affinity DataIC50:  9nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354791(CHEMBL1834471)
Affinity DataIC50:  9nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354783(CHEMBL1834463)
Affinity DataIC50:  10nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354794(CHEMBL1834474)
Affinity DataIC50:  10nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354793(CHEMBL1834473)
Affinity DataIC50:  10nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354790(CHEMBL1834470)
Affinity DataIC50:  11nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354802(CHEMBL1834482)
Affinity DataIC50:  11nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354801(CHEMBL1834481)
Affinity DataIC50:  13nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354784(CHEMBL1834464)
Affinity DataIC50:  14nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354795(CHEMBL1834475)
Affinity DataIC50:  15nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354787(CHEMBL1834467)
Affinity DataIC50:  16nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  16nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354785(CHEMBL1834465)
Affinity DataIC50:  17nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354798(CHEMBL1834478)
Affinity DataIC50:  17nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50354796(CHEMBL1834476)
Affinity DataIC50:  18nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  290nMAssay Description:Inhibition of HDAC1 by fluorescent activity assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  368nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  500nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  501nMAssay Description:Inhibition of HDAC3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385017(CHEMBL2035393)
Affinity DataIC50:  700nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385007(CHEMBL2035382)
Affinity DataIC50:  900nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385015(CHEMBL2035390)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385004(CHEMBL2035379)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385021(CHEMBL2035392)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385012(CHEMBL2035387)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385001(CHEMBL2034986)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385003(CHEMBL2035378)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385016(CHEMBL2035391)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385006(CHEMBL2035381)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385014(CHEMBL2035389)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385002(CHEMBL2035377)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385013(CHEMBL2035388)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385005(CHEMBL2035380)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385018(CHEMBL2035394)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385008(CHEMBL2035383)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385019(CHEMBL2035395)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385011(CHEMBL2035386)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385009(CHEMBL2035384)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385020(CHEMBL2035396)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385010(CHEMBL2035385)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM50385000(CHEMBL2035376)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of HDAC1 using Fluor de Lys as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Guru Ghasidas University

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of HDAC4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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