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Found 84 with Last Name = 'rajendran' and Initial = 'p'
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65470(Quinolone-based HDAC inhibitor 4i)
Affinity DataIC50:  0.100nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65471(Quinolone-based HDAC inhibitor 4j)
Affinity DataIC50:  1.5nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65478(Quinolone-based HDAC inhibitor 4o)
Affinity DataIC50:  10nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97708(US8476255, 96)
Affinity DataIC50:  10nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97707(US8476255, 95)
Affinity DataIC50:  10nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143215(CHEMBL3758457)
Affinity DataIC50:  16nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97695(US8476255, 55)
Affinity DataIC50:  20nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 6(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  23nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistone deacetylase 3(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143215(CHEMBL3758457)
Affinity DataIC50:  25nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143215(CHEMBL3758457)
Affinity DataIC50:  27nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65481(Quinolone-based HDAC inhibitor 4r)
Affinity DataIC50:  28nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65479(Quinolone-based HDAC inhibitor 4p)
Affinity DataIC50:  28nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97703(US8476255, 89)
Affinity DataIC50:  30nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97698(US8476255, 59)
Affinity DataIC50:  30nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65475(Quinolone-based HDAC inhibitor 4l)
Affinity DataIC50:  32nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65474(Quinolone-based HDAC inhibitor 4k)
Affinity DataIC50:  32nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65458(Quinolone-based HDAC inhibitor 4a)
Affinity DataIC50:  32nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97685(US8476255, 28)
Affinity DataIC50:  36nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 3(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  38nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65485(Quinolone-based HDAC inhibitor 4v)
Affinity DataIC50:  39nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65463(Quinolone-based HDAC inhibitor 4c)
Affinity DataIC50:  39nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97704(US8476255, 90)
Affinity DataIC50:  40nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97694(US8476255, 53)
Affinity DataIC50:  40nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97697(US8476255, 58)
Affinity DataIC50:  40nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65480(Quinolone-based HDAC inhibitor 4q)
Affinity DataIC50:  40nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97706(US8476255, 94)
Affinity DataIC50:  40nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143215(CHEMBL3758457)
Affinity DataIC50:  42nMAssay Description:Inhibition of HDAC10 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65469(Quinolone-based HDAC inhibitor 4h)
Affinity DataIC50:  42nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97680(US8476255, 19)
Affinity DataIC50:  42nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  43nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  45nMAssay Description:Inhibition of human HDAC8More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97700(US8476255, 77)
Affinity DataIC50:  50nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97684(US8476255, 27)
Affinity DataIC50:  50nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97688(US8476255, 32)
Affinity DataIC50:  52nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97687(US8476255, 31)
Affinity DataIC50:  54nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 2(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143215(CHEMBL3758457)
Affinity DataIC50:  54nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97686(US8476255, 29)
Affinity DataIC50:  57nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97701(US8476255, 84)
Affinity DataIC50:  60nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97699(BOC-LYS(AC)-AMC | US8476255, 76)
Affinity DataIC50:  60nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97693(US8476255, 52)
Affinity DataIC50:  60nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97683(US8476255, 24)
Affinity DataIC50:  62nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  64nMAssay Description:Inhibition of HDAC10 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97696(US8476255, 57)
Affinity DataIC50:  70nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97709(US8476255, 101)
Affinity DataIC50:  70nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65476(Quinolone-based HDAC inhibitor 4m)
Affinity DataIC50:  75nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65484(Quinolone-based HDAC inhibitor 4u)
Affinity DataIC50:  85nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Npo-International Laboratory Of Biochemistry

Curated by ChEMBL
LigandPNGBDBM50241294(CHEMBL240954 | SL-0101 | kaempferol 3-O-(3'',4''-d...)
Affinity DataIC50:  89nMAssay Description:Inhibition of his-tagged active RSK2 (unknown origin) expressed in Sf9 cells after 10 to 45 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65468(Quinolone-based HDAC inhibitor 4g)
Affinity DataIC50:  90nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM65472(Quinolone-based HDAC inhibitor 4w)
Affinity DataIC50:  95nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1/11/4/6/8(Homo sapiens (Human))
Orchid Chemicals & Pharmaceuticals

LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  110nMAssay Description:Histone Deacetylase (HDAC) Inhibition Assay using Boc-Lys(Ac)-AMC Substrate: Inhibition of HDAC has been implicated to modulate transcription and to ...More data for this Ligand-Target Pair
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