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Found 181 with Last Name = 'rehman' and Initial = 'a'
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50275870(CHEMBL4129331)
Affinity DataKi:  115nMAssay Description:Mixed-type inhibition of calf intestinal alkaline phosphatase assessed as enzyme-inhibitor dissociation constant using varying levels of p-NPP as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50275870(CHEMBL4129331)
Affinity DataKi:  415nMAssay Description:Mixed-type inhibition of calf intestinal alkaline phosphatase assessed as enzyme-substrate-inhibitor dissociation constant using varying levels of p-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435064(CHEMBL2391315)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325684((S)-2-((4R,5R)-5-(biphenyl-2-ylcarbamoyl)-1,3-diox...)
Affinity DataIC50:  100nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435063(CHEMBL2391316)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
Universiti Teknologi Mara (Uitm), Puncak Alam Campus

LigandPNGBDBM60585(2-(3'-Fluorophenyl)-7-methyl-1H-benzo[d]imidazole ...)
Affinity DataIC50:  165nMAssay Description:The 135 µL of 50 mM phosphate saline buffer pH (6.8), solution of enzyme (20 µL), and 20 µL of test sample with 70% DMSO was added to 96-well plate. ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325710((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  200nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50275870(CHEMBL4129331)
Affinity DataIC50:  251nMAssay Description:Inhibition of calf intestinal alkaline phosphatase using p-NPP as substrate pretreated for 10 mins followed by substrate addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435079(CHEMBL2391321)
Affinity DataIC50:  290nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325699((S)-2-((4R,5R)-5-(cyclopropylcarbamoyl)-1,3-dioxol...)
Affinity DataIC50:  300nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50275871(CHEMBL4128234)
Affinity DataIC50:  344nMAssay Description:Inhibition of calf intestinal alkaline phosphatase using p-NPP as substrate pretreated for 10 mins followed by substrate addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435078(CHEMBL2391322)
Affinity DataIC50:  370nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325714((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  400nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435070(CHEMBL2391499)
Affinity DataIC50:  430nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50275925(CHEMBL4130271)
Affinity DataIC50:  492nMAssay Description:Inhibition of calf intestinal alkaline phosphatase using p-NPP as substrate pretreated for 10 mins followed by substrate addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325712((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  500nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325689((S)-2-((4R,5R)-5-(biphenyl-2-ylcarbamoyl)-1,3-diox...)
Affinity DataIC50:  500nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325707((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  600nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325700((S)-2-((4R,5R)-5-(benzo[d]thiazol-2-ylcarbamoyl)-1...)
Affinity DataIC50:  600nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325702((S)-2-((4R,5R)-5-(2-(1H-indol-3-yl)ethylcarbamoyl)...)
Affinity DataIC50:  600nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325704((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  600nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435077(CHEMBL2391323)
Affinity DataIC50:  690nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325701((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  700nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325713((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  700nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325705((S)-2-((4R,5R)-5-(2-chlorophenylcarbamoyl)-1,3-dio...)
Affinity DataIC50:  700nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435069(CHEMBL2391310)
Affinity DataIC50:  760nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435062(CHEMBL2391317)
Affinity DataIC50:  830nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435067(CHEMBL2391312)
Affinity DataIC50:  890nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50275869(CHEMBL4126012)
Affinity DataIC50:  896nMAssay Description:Inhibition of calf intestinal alkaline phosphatase using p-NPP as substrate pretreated for 10 mins followed by substrate addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325709((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  900nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435068(CHEMBL2391311)
Affinity DataIC50:  980nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325715((S)-2-((4R,5R)-5-(1-benzyl-3-tert-butyl-1H-pyrazol...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325694((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325698((S)-2-((4R,5R)-5-(tert-butylcarbamoyl)-1,3-dioxola...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435076(CHEMBL2391493)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325691((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435058(CHEMBL2391309)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435075(CHEMBL2391494)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435066(CHEMBL2391313)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325690((S)-2-((4R,5R)-5-(cyclohexylcarbamoyl)-1,3-dioxola...)
Affinity DataIC50:  1.40E+3nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325708((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325693((S)-2-((4R,5R)-5-(butylcarbamoyl)-1,3-dioxolane-4-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435061(CHEMBL2391318)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325711((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
New Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50325696((S)-3-(4-(2,6-dichlorobenzyloxy)phenyl)-2-((4R,5R)...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of VCAM1 from VLA4 receptor in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50275874(CHEMBL4125873)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of calf intestinal alkaline phosphatase using p-NPP as substrate pretreated for 10 mins followed by substrate addition measured after 30 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50275882(CHEMBL4126859)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibition of calf intestinal alkaline phosphatase using p-NPP as substrate pretreated for 10 mins followed by substrate addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50275883(CHEMBL4126997)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of calf intestinal alkaline phosphatase using p-NPP as substrate pretreated for 10 mins followed by substrate addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435074(CHEMBL2391495)
Affinity DataIC50:  1.80E+3nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50435073(CHEMBL2391496)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist activity at VLA-4 receptor in human U937 cells assessed as inhibition of VCAM-1 binding by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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