TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged C-terminal His6-tagged MEK1 expressed in Escherichia coli using myelin basic protei...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged C-terminal His6-tagged MEK1 expressed in Escherichia coli using myelin basic protei...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of MEK1 in BRAF mutant human A549 cells assessed as reduction in ERK1/2 phosphorylation by ELISAMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 3.12E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 6.57E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 7.22E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 8.03E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 9.08E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 9.36E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of FAK in human MCF7 cellsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.91E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 2.63E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 2.72E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 3.46E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 3.83E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 4.06E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair