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Found 40 with Last Name = 'ren' and Initial = 'zl'
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
Affinity DataIC50:  89nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged C-terminal His6-tagged MEK1 expressed in Escherichia coli using myelin basic protei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50536790(CHEMBL4575118)
Affinity DataIC50:  91nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged C-terminal His6-tagged MEK1 expressed in Escherichia coli using myelin basic protei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137968(CHEMBL3754002)
Affinity DataIC50:  280nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataIC50:  570nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50536790(CHEMBL4575118)
Affinity DataIC50:  610nMAssay Description:Inhibition of MEK1 in BRAF mutant human A549 cells assessed as reduction in ERK1/2 phosphorylation by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137968(CHEMBL3754002)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137851(CHEMBL3752866)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137701(CHEMBL3752369)
Affinity DataIC50:  1.74E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137701(CHEMBL3752369)
Affinity DataIC50:  3.12E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138037(CHEMBL3752051)
Affinity DataIC50:  6.57E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM12915(2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one |...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137851(CHEMBL3752866)
Affinity DataIC50:  7.22E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137967(CHEMBL3752088)
Affinity DataIC50:  8.03E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50536790(CHEMBL4575118)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137656(CHEMBL3753671)
Affinity DataIC50:  9.08E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137685(CHEMBL3753973)
Affinity DataIC50:  9.36E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138037(CHEMBL3752051)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137685(CHEMBL3753973)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137967(CHEMBL3752088)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137656(CHEMBL3753671)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50536790(CHEMBL4575118)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of FAK in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138034(CHEMBL3752413)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138021(CHEMBL3752400)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138042(CHEMBL3752044)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137952(CHEMBL3753798)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138036(CHEMBL3752641)
Affinity DataIC50:  1.91E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137970(CHEMBL3754379)
Affinity DataIC50:  2.02E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137969(CHEMBL3753152)
Affinity DataIC50:  2.02E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138031(CHEMBL3753037)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138032(CHEMBL3754182)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50536790(CHEMBL4575118)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50536790(CHEMBL4575118)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50536790(CHEMBL4575118)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138024(CHEMBL3754755)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138022(CHEMBL3752335)
Affinity DataIC50:  2.63E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137971(CHEMBL3753949)
Affinity DataIC50:  2.72E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138030(CHEMBL3754381)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138031(CHEMBL3753037)
Affinity DataIC50:  3.46E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138032(CHEMBL3754182)
Affinity DataIC50:  3.83E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138024(CHEMBL3754755)
Affinity DataIC50:  4.06E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed