Affinity DataKi: 6nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory activity against bovine coagulation factor X expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Institut FüR Biochemie
Curated by ChEMBL
Institut FüR Biochemie
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibitory activity against human tissue-type plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Compound was tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Inhibitory activity against bovine coagulation factor X expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Compound was tested for inhibition of plasminMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Tested for inhibition of plasminMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Institut FüR Biochemie
Curated by ChEMBL
Institut FüR Biochemie
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Inhibitory activity against human urokinase plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Institut FüR Biochemie
Curated by ChEMBL
Institut FüR Biochemie
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Compound was tested for inhibition of plasminogen activator urokinase(microPa)More data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Compound was tested for inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair