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Found 89 with Last Name = 'robertus' and Initial = 'jd'
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
The University of Texas

LigandPNGBDBM50138983((S)-2-Amino-5-(2-methyl-isothioureido)-pentanoic a...)
Affinity DataKi:  50nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
The University of Texas

LigandPNGBDBM92901(ADMA, 3)
Affinity DataKi:  700nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
The University of Texas

LigandPNGBDBM50072297((S)-5-Acetimidoylamino-2-amino-pent | (S)-5-Acetim...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM92900(CHEMBL1835117 | L-Arginine, 2 | NMMA, 2)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
The University of Texas

LigandPNGBDBM50254450((S)-2-Amino-5-propionimidoylamino-pentanoic acid |...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN(G),N(G)-dimethylarginine dimethylaminohydrolase 1(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM92904(nNOS and DDAH inhibitor, 14)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetNitric oxide synthase, brain(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM92904(nNOS and DDAH inhibitor, 14)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN(G),N(G)-dimethylarginine dimethylaminohydrolase 1(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM50254450((S)-2-Amino-5-propionimidoylamino-pentanoic acid |...)
Affinity DataKi:  5.20E+4nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
TargetN(G),N(G)-dimethylarginine dimethylaminohydrolase 1(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM92905(DDAH Inhibitor, 15)
Affinity DataKi:  1.10E+5nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN(G),N(G)-dimethylarginine dimethylaminohydrolase 1(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM92900(CHEMBL1835117 | L-Arginine, 2 | NMMA, 2)
Affinity DataKi:  1.31E+5nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN(G),N(G)-dimethylarginine dimethylaminohydrolase 1(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM92900(CHEMBL1835117 | L-Arginine, 2 | NMMA, 2)
Affinity DataKi:  2.90E+5nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN(G),N(G)-dimethylarginine dimethylaminohydrolase 1(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM50072297((S)-5-Acetimidoylamino-2-amino-pent | (S)-5-Acetim...)
Affinity DataKi:  9.90E+5nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
The University of Texas

LigandPNGBDBM92903(L-Citrulline, 4)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN(G),N(G)-dimethylarginine dimethylaminohydrolase 1(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM92900(CHEMBL1835117 | L-Arginine, 2 | NMMA, 2)
Affinity DataKi:  1.20E+6nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN(G),N(G)-dimethylarginine dimethylaminohydrolase 1(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM92900(CHEMBL1835117 | L-Arginine, 2 | NMMA, 2)
Affinity DataKi:  1.40E+6nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
The University of Texas

LigandPNGBDBM92905(DDAH Inhibitor, 15)
Affinity DataKi: >1.90E+6nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN(G),N(G)-dimethylarginine dimethylaminohydrolase 1(Homo sapiens (Human))
The University of Texas

LigandPNGBDBM92903(L-Citrulline, 4)
Affinity DataKi:  3.70E+6nMAssay Description:Inhibition assay using DDAH-1 and nNOS.More data for this Ligand-Target Pair
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424241(CHEMBL2314138)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50420411(CHEMBL2089319)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Ricinus communis ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424235(CHEMBL2314130)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424238(CHEMBL2314127)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424242(CHEMBL2314137)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424239(CHEMBL2314140)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424231(CHEMBL2314134)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424234(CHEMBL2314131)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445065(CHEMBL3098919)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445071(CHEMBL3098913)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50420407(CHEMBL2089314)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of Ricinus communis ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424233(CHEMBL2314132)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424232(CHEMBL2314133)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445069(CHEMBL3098915)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445068(CHEMBL3098916)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424240(CHEMBL2314139)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445073(CHEMBL3098911)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445072(CHEMBL3098912)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445070(CHEMBL3098914)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445075(CHEMBL3098909)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424229(CHEMBL2314136)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424230(CHEMBL2314135)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445063(CHEMBL3098907)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50420404(CHEMBL2089311)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of Ricinus communis ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445074(CHEMBL3098910)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424237(CHEMBL2314128)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424228(CHEMBL2311565)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50420410(CHEMBL2089318)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of Ricinus communis ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50424236(CHEMBL2314129)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of Ricin toxin A after 90 mins by luciferase-translational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445076(CHEMBL3098908)
Affinity DataIC50:  1.28E+5nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50420413(CHEMBL2089310)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of Ricinus communis ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50420415(CHEMBL2086423)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of Ricinus communis ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRicin(Ricinus communis)
Toho University

Curated by ChEMBL
LigandPNGBDBM50445064(CHEMBL3098906)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of castor bean ricin toxin A after 90 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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