Affinity DataKi: 1nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity for Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity for Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 206nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 753nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+4nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+4nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 3.50E+4nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 6.50E+4nMAssay Description:Binding affinity was measured on Cytochrome P450 19A1More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Homo sapiens (Human))
University of North Carolina
University of North Carolina
Affinity DataIC50: 0.300nMpH: 7.5 T: 2°CAssay Description:Enzymatic activities were assayed using [3H] cAMP and [3H]cGMP as substrate.More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University of North Carolina At Chapel Hill
University of North Carolina At Chapel Hill
Affinity DataIC50: 0.400nMpH: 7.5 T: 2°CAssay Description:PDE4 catalytic activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using PDE-SPA kit (Amersham International). [3H]-AMP was c...More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University of North Carolina At Chapel Hill
University of North Carolina At Chapel Hill
Affinity DataIC50: 0.400nMpH: 7.5 T: 2°CAssay Description:PDE4 catalytic activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using PDE-SPA kit (Amersham International). [3H]-AMP was c...More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
University of North Carolina At Chapel Hill
University of North Carolina At Chapel Hill
Affinity DataIC50: 0.400nMpH: 7.5 T: 2°CAssay Description:PDE4 catalytic activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using PDE-SPA kit (Amersham International). [3H]-AMP was c...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Research And Development Laboratories
Curated by ChEMBL
Research And Development Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.510nMAssay Description:Compound was tested for inhibitory activity against angiotensin I converting enzymeMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Research And Development Laboratories
Curated by ChEMBL
Research And Development Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Compound was tested for inhibitory activity against angiotensin I converting enzymeMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Research And Development Laboratories
Curated by ChEMBL
Research And Development Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Compound was tested for inhibitory activity against angiotensin I converting enzymeMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Research And Development Laboratories
Curated by ChEMBL
Research And Development Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Compound was tested for inhibitory activity against angiotensin I converting enzymeMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Homo sapiens (Human))
University of North Carolina At Chapel Hill
University of North Carolina At Chapel Hill
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:PDE4 catalytic activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using PDE-SPA kit (Amersham International). [3H]-AMP was c...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Research And Development Laboratories
Curated by ChEMBL
Research And Development Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Compound was tested for inhibitory activity against angiotensin I converting enzymeMore data for this Ligand-Target Pair