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Found 796 with Last Name = 'romero' and Initial = 'j'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  0.280nMAssay Description:Agonist activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidad De M£Laga

Curated by ChEMBL
LigandPNGBDBM50308567(CHEMBL592891 | N-(4-acetylphenyl)-2-(4-(7-methyl-2...)
Affinity DataKi:  1.39nMAssay Description:Inhibition of adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  1.90nMAssay Description:Agonist activity at CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidad De M£Laga

Curated by ChEMBL
LigandPNGBDBM50004566(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinaz...)
Affinity DataKi:  2.27nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in in human HeLa cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidad De M£Laga

Curated by ChEMBL
LigandPNGBDBM50053929(CHEMBL88147 | N-(9-Chloro-2-furan-2-yl-[1,2,4]tria...)
Affinity DataKi:  2.48nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in human HeLa cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidad De M£Laga

Curated by ChEMBL
LigandPNGBDBM50308566(8-(4-(3,6,9,12-tetraoxatricos-22-enyloxy)phenyl)-t...)
Affinity DataKi:  4.16nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidad De M£Laga

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  19.3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidad De M£Laga

Curated by ChEMBL
LigandPNGBDBM50308568(2-(2-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKi:  23.2nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO-A1 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50160434((6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-indol-3-...)
Affinity DataKi:  31nMAssay Description:Inverse agonist activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  40nMAssay Description:Agonist activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  40nMAssay Description:Agonist activity at CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207242(CHEMBL3901140)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207259(CHEMBL3892181)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207267(CHEMBL3960083)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207271(CHEMBL594935)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidad De M£Laga

Curated by ChEMBL
LigandPNGBDBM50308566(8-(4-(3,6,9,12-tetraoxatricos-22-enyloxy)phenyl)-t...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in in human HeLa cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207256(CHEMBL3898407)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207261(CHEMBL3891003)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207255(CHEMBL3944807)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207239(CHEMBL3907898)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207269(CHEMBL3907434)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207254(CHEMBL3938131)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207247(CHEMBL3920181)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207266(CHEMBL3932295)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207257(CHEMBL3950235)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207244(CHEMBL3916891)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207255(CHEMBL3944807)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207258(CHEMBL3889952)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207245(CHEMBL3898882)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207240(CHEMBL3917967)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207263(CHEMBL3922512)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207271(CHEMBL594935)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM106773(2‐(4‐methoxyphenyl)‐1‐[(4&...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207244(CHEMBL3916891)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207250(CHEMBL3915743)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207241(CHEMBL3895577)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207262(CHEMBL3898880)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207258(CHEMBL3889952)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207251(CHEMBL3916164)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207265(CHEMBL3914550)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207270(CHEMBL3926929)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207248(CHEMBL3904520)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207252(CHEMBL3935866)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207260(CHEMBL3905573)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207246(CHEMBL3984372)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidad De M£Laga

Curated by ChEMBL
LigandPNGBDBM10847(1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dion...)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207251(CHEMBL3916164)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207254(CHEMBL3938131)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207267(CHEMBL3960083)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207246(CHEMBL3984372)
Affinity DataKi:  4.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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