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Found 182 with Last Name = 'romero' and Initial = 'ja'
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501754(CHEMBL4071396)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501764(CHEMBL4061199)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 847More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501755(CHEMBL4077947)
Affinity DataIC50:  1nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501762(CHEMBL4081478)
Affinity DataIC50:  1nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501782(CHEMBL4087371)
Affinity DataIC50:  1nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200120(CHEMBL260091 | CHIR-090 | US10875832, Compound ChI...)
Affinity DataIC50: <1nMAssay Description:Displacement of fluorescent ligand from Pseudomonas aeruginosa LpxC measured after 30 mins by fluorescence anisotrophy assayMore data for this Ligand-Target Pair
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501780(CHEMBL4083988)
Affinity DataIC50:  1nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 847More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501779(CHEMBL4102207)
Affinity DataIC50:  1nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501764(CHEMBL4061199)
Affinity DataIC50:  1nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501756(CHEMBL4066982)
Affinity DataIC50:  2nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501768(CHEMBL4102818)
Affinity DataIC50:  2nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501753(CHEMBL4098438)
Affinity DataIC50:  2nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 847More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501780(CHEMBL4083988)
Affinity DataIC50:  2nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501754(CHEMBL4071396)
Affinity DataIC50:  2nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501778(CHEMBL4098674)
Affinity DataIC50:  2nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501770(CHEMBL4092719)
Affinity DataIC50:  2nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 847More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501753(CHEMBL4098438)
Affinity DataIC50:  2nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501752(CHEMBL4095059)
Affinity DataIC50:  2nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501764(CHEMBL4061199)
Affinity DataIC50:  3nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501783(CHEMBL4064896)
Affinity DataIC50:  3nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501761(CHEMBL4068010)
Affinity DataIC50:  3nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501753(CHEMBL4098438)
Affinity DataIC50:  3nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501767(CHEMBL4091763)
Affinity DataIC50:  3nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501762(CHEMBL4081478)
Affinity DataIC50:  4nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501752(CHEMBL4095059)
Affinity DataIC50:  4nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501770(CHEMBL4092719)
Affinity DataIC50:  4nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50173889(CHEMBL3809400)
Affinity DataIC50:  4nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseB ATPase activity using linear pBR322 DNA substrate incubated for 30 mins by fluorescence polarization ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501770(CHEMBL4092719)
Affinity DataIC50:  4nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501782(CHEMBL4087371)
Affinity DataIC50:  5nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501766(CHEMBL4070896)
Affinity DataIC50:  5nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501763(CHEMBL4099505)
Affinity DataIC50:  5nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501763(CHEMBL4099505)
Affinity DataIC50:  5nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501767(CHEMBL4091763)
Affinity DataIC50:  5nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501761(CHEMBL4068010)
Affinity DataIC50:  5nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501780(CHEMBL4083988)
Affinity DataIC50:  6nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501786(CHEMBL4089353)
Affinity DataIC50:  6nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50173875(CHEMBL3808756)
Affinity DataIC50:  6nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseB ATPase activity using linear pBR322 DNA substrate incubated for 30 mins by fluorescence polarization ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50173879(CHEMBL3810359)
Affinity DataIC50:  6nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseB ATPase activity using linear pBR322 DNA substrate incubated for 30 mins by fluorescence polarization ...More data for this Ligand-Target Pair
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501755(CHEMBL4077947)
Affinity DataIC50:  6nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501779(CHEMBL4102207)
Affinity DataIC50:  6nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501760(CHEMBL4078871)
Affinity DataIC50:  6nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501775(CHEMBL4077504)
Affinity DataIC50:  7nMAssay Description:Inhibition of LpxC in Escherichia coli isolate 35 ATCC 25922More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50173641(CHEMBL3810223)
Affinity DataIC50:  8nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseB ATPase activity using linear pBR322 DNA substrate incubated for 30 mins by fluorescence polarization ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501766(CHEMBL4070896)
Affinity DataIC50:  8nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50134212(CHEMBL3741453)
Affinity DataIC50: <8nMAssay Description:Inhibition of Staphylococcus aureus Gyrase B ATPase activity by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50173644(CHEMBL3810048)
Affinity DataIC50: <8nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseB ATPase activity using linear pBR322 DNA substrate incubated for 30 mins by fluorescence polarization ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50499015(CHEMBL3736321)
Affinity DataIC50:  8nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50173857(CHEMBL3808789)
Affinity DataIC50: <8nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseB ATPase activity using linear pBR322 DNA substrate incubated for 30 mins by fluorescence polarization ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50173823(CHEMBL3809278)
Affinity DataIC50:  8nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseB ATPase activity using linear pBR322 DNA substrate incubated for 30 mins by fluorescence polarization ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50501783(CHEMBL4064896)
Affinity DataIC50:  8nMAssay Description:Inhibition of LpxC in Pseudomonas aeruginosa isolate 44 ATCC 27853More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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