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Found 205 with Last Name = 'rosenblum' and Initial = 'js'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50050517(Boronic acid derivative | CHEMBL305170 | N-alkyl G...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171546((S)-2,4-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...)
Affinity DataIC50:  0.480nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50196928((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of human DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  0.720nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171653(CHEMBL196120 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50196929((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...)
Affinity DataIC50:  0.880nMAssay Description:Inhibition of human DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataIC50:  0.890nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171648(CHEMBL372180 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171649(CHEMBL196933 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171645(2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50:  2.20nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171558(2,6-Diamino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  3.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171650(2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171656(2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50:  4.10nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  4.5nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171647(CHEMBL373269 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  4.60nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  4.60nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171553(2,5-Diamino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  4.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM15234((1R,3R,5S,9R,18S)-18-(methoxymethyl)-1,5-dimethyl-...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of AX7503 binding to recombinant Plk1 (unknown origin) by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171653(CHEMBL196120 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  6.30nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  6.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171649(CHEMBL196933 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  7.80nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171657(2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171647(CHEMBL373269 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171559((S)-2,3-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...)
Affinity DataIC50:  8.20nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against human fibroblast activation protein alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050517(Boronic acid derivative | CHEMBL305170 | N-alkyl G...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50354779(CHEMBL1834330)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant full length GSK3beta after 1 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171644(CHEMBL427012 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50354765(CHEMBL1834315)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant full length GSK3beta after 1 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171651(2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171551((S)-2-Amino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  18nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50354767(CHEMBL1834318)
Affinity DataIC50:  22nMAssay Description:Inhibition of human recombinant full length GSK3beta after 1 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171657(2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171651(2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171650(2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50171656(2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  30nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50354773(CHEMBL1834324)
Affinity DataIC50:  31nMAssay Description:Inhibition of human recombinant full length GSK3beta after 1 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50354764(CHEMBL1834125)
Affinity DataIC50:  31nMAssay Description:Inhibition of human recombinant full length GSK3beta after 1 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171652(CHEMBL381444 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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