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Found 24 with Last Name = 'rotolo' and Initial = 'c'
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  90nMAssay Description:Inhibition of recombinant human PDE4D3 expressed in baculoviral systemMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50057795(CHEMBL3326090)
Affinity DataIC50:  210nMAssay Description:Inhibition of recombinant human PDE4D3 expressed in baculoviral systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50057791(CHEMBL3326083)
Affinity DataIC50:  660nMAssay Description:Inhibition of recombinant human PDE4D3 expressed in baculoviral systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50057794(CHEMBL3326089)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of recombinant human PDE4D3 expressed in baculoviral systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50057792(CHEMBL3326084)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of recombinant human PDE4D3 expressed in baculoviral systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50057791(CHEMBL3326083)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of PDE4B2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50057793(CHEMBL3326087)
Affinity DataIC50:  1.79E+3nMAssay Description:Inhibition of recombinant human PDE4D3 expressed in baculoviral systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50299569(3-(cyclopentyloxy)-4-methoxybenzaldehyde O-[2-(2,6...)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of recombinant human PDE4D3 expressed in baculoviral systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493837(CHEMBL2443298)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493837(CHEMBL2443298)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493838(CHEMBL2443297)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493835(CHEMBL2443288)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493846(CHEMBL2443290)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50299568(3-(Cyclopentyloxy)-4-methoxybenzaldehyde O-[3-(2,6...)
Affinity DataIC50:  3.46E+3nMAssay Description:Inhibition of recombinant human PDE4D3 expressed in baculoviral systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50057795(CHEMBL3326090)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of PDE4B2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM241949(US9428466, Merbarone)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493842(CHEMBL2443291)
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493841(CHEMBL2443289)
Affinity DataIC50: >3.50E+4nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493836(CHEMBL2443299)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493845(CHEMBL2443300)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493843(CHEMBL2443296)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493844(CHEMBL2440361)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493840(CHEMBL2440360)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50493839(CHEMBL2443292)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed