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Found 294 with Last Name = 'ruan' and Initial = 'bf'
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  100nMAssay Description:Inhibition of COX-2 (unknown origin) by chemiluminescence assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  120nMAssay Description:Inhibition of COX2 by chemiluminescent enzyme assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  120nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429262(CHEMBL2334141)
Affinity DataIC50:  280nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429284(CHEMBL2333743)
Affinity DataIC50:  390nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429285(CHEMBL2333742)
Affinity DataIC50:  450nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429271(CHEMBL2333735)
Affinity DataIC50:  460nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50575103(CHEMBL4849582)
Affinity DataIC50:  560nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-stimulated mouse bone marrow-derived macrophages assessed as reduction in IL-1beta secretion prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429273(CHEMBL2333733)
Affinity DataIC50:  580nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429282(CHEMBL2333745)
Affinity DataIC50:  720nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50575102(CHEMBL4870161)
Affinity DataIC50:  760nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-stimulated mouse bone marrow-derived macrophages assessed as reduction in IL-1beta secretion prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50357965(CHEMBL1916969)
Affinity DataIC50:  800nMAssay Description:Inhibition of COX2 by chemiluminescent enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50575106(Ent-Oridonin | Oridonin)
Affinity DataIC50:  810nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-stimulated mouse bone marrow-derived macrophages assessed as reduction in IL-1beta secretion prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605174(CHEMBL1164920)
Affinity DataIC50:  810nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429268(CHEMBL2333738)
Affinity DataIC50:  850nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237225(1-(4-Bromophenyl)-1-(4-hydroxy-3-methoxybenzyl)-3-...)
Affinity DataIC50:  970nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429262(CHEMBL2334141)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of COX-2 (unknown origin) by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605172(CHEMBL5202921)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetETS domain-containing protein Elk-1(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237214(1-(4-Bromophenyl)-1-(4-hydroxy-3-methoxybenzyl)-3-...)
Affinity DataIC50:  1.24E+3nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1/3(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237225(1-(4-Bromophenyl)-1-(4-hydroxy-3-methoxybenzyl)-3-...)
Affinity DataIC50:  1.27E+3nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429284(CHEMBL2333743)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of COX-2 (unknown origin) by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429285(CHEMBL2333742)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of COX-2 (unknown origin) by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50575101(CHEMBL4852097)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-stimulated mouse bone marrow-derived macrophages assessed as reduction in IL-1beta secretion prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237214(1-(4-Bromophenyl)-1-(4-hydroxy-3-methoxybenzyl)-3-...)
Affinity DataIC50:  1.38E+3nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50575104(CHEMBL4852880)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-stimulated mouse bone marrow-derived macrophages assessed as reduction in IL-1beta secretion prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429271(CHEMBL2333735)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of COX-2 (unknown origin) by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetETS domain-containing protein Elk-1(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237225(1-(4-Bromophenyl)-1-(4-hydroxy-3-methoxybenzyl)-3-...)
Affinity DataIC50:  1.53E+3nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605166(CHEMBL5179667)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429269(CHEMBL2333737)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429268(CHEMBL2333738)
Affinity DataIC50:  1.88E+3nMAssay Description:Inhibition of COX-2 (unknown origin) by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50357967(CHEMBL1916968)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of COX2 by chemiluminescent enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237222(1-(4-Hydroxy-3-methoxybenzyl)-1-(4-methoxyphenyl)-...)
Affinity DataIC50:  1.93E+3nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetETS domain-containing protein Elk-1(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237223(1-(4-Fluorophenyl)-1-(4-hydroxy-3-methoxybenzyl)-3...)
Affinity DataIC50:  1.95E+3nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429273(CHEMBL2333733)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibition of COX-2 (unknown origin) by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429277(CHEMBL2333750)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429282(CHEMBL2333745)
Affinity DataIC50:  2.01E+3nMAssay Description:Inhibition of COX-2 (unknown origin) by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429263(CHEMBL2334140)
Affinity DataIC50:  2.08E+3nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429279(CHEMBL2333748)
Affinity DataIC50:  2.09E+3nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429296(CHEMBL2333753)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1/3(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237214(1-(4-Bromophenyl)-1-(4-hydroxy-3-methoxybenzyl)-3-...)
Affinity DataIC50:  2.14E+3nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605173(CHEMBL5195047)
Affinity DataIC50:  2.15E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429294(CHEMBL2333755)
Affinity DataIC50:  2.15E+3nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50155928(3,4-Methylenedioxyb-Nitrostyrene | CHEMBL596380)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50155928(3,4-Methylenedioxyb-Nitrostyrene | CHEMBL596380)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-stimulated mouse bone marrow-derived macrophages assessed as reduction in IL-1beta secretion prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetETS domain-containing protein Elk-1(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237222(1-(4-Hydroxy-3-methoxybenzyl)-1-(4-methoxyphenyl)-...)
Affinity DataIC50:  2.42E+3nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429276(CHEMBL2334136)
Affinity DataIC50:  2.44E+3nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetETS domain-containing protein Elk-1(Homo sapiens (Human))
Nanjing University

LigandPNGBDBM237224(1-(4-Chlorophenyl)-1-(4-hydroxy-3-methoxybenzyl)-3...)
Affinity DataIC50:  2.47E+3nMAssay Description:Detection of the effect of compounds on p-MEK1/2, t-ERK1/2, pERK1/2, p-Rsk1 and p-Elk-1 activity in B16-F10 cells was performed using ELISA kits (Inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50429291(CHEMBL2334131)
Affinity DataIC50:  2.56E+3nMAssay Description:Inhibition of COX-2 in mouse RAW264.7 cells assessed as decrease in LPS-induced PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM50357964(CHEMBL1916967)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of COX2 by chemiluminescent enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50105463(2,7-diamino-10-ethyl-9-phenylphenanthridinium brom...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of telomerase activity expressed in human SGC7901 cells by SYBER green dye based TRAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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