Affinity DataKi: 0.146nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.226nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.257nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.268nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Displacement of [3H]-aldosterone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.342nMAssay Description:Displacement of [3H]-aldosterone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Displacement of [3H]-aldosterone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.967nMAssay Description:Displacement of [3H]-aldosterone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-aldosterone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]-methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]-aldosterone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]-methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Displacement of [3H]-methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [3H]-methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Displacement of [3H]-methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [3H]-dexamethasone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 239nMAssay Description:Displacement of [3H]-methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 418nMAssay Description:Displacement of [3H]-methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 561nMAssay Description:Displacement of [3H]-methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.41E+3nMAssay Description:Displacement of [3H]-methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.52E+3nMAssay Description:Displacement of [3H]-methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Binding affinity to BRPF3 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of human ATAD2A (981 to 1108 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Target4-hydroxyphenylpyruvate dioxygenase(Homo sapiens (Human))
Central China Normal University
Curated by ChEMBL
Central China Normal University
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant His-tagged HPPD expressed in Escherichia coli BL21(DE3) by UV/visible plate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of human BRPF1 (627 to 740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair