Affinity DataIC50: 0.100nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.380nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.420nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.510nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.510nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.610nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.690nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.740nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.770nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.840nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.990nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of LPS stimulated TNF alpha release in whole bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.87nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of LPS stimulated TNF alpha release in whole bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.59nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of LPS stimulated TNF alpha release in whole bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 3.32nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.75nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of TNF alpha release in THP1 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of DiTc binding to Kv1.3 channel in human brain membranesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of DiTc binding to Kv1.3 channel in human brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of LPS stimulated TNF alpha release in whole bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Inhibition of LPS stimulated TNF alpha release in whole bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Inhibition of LPS stimulated TNF alpha release in whole bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Inhibition of LPS stimulated TNF alpha release in whole bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: 7.71nMAssay Description:Inhibition of LPS stimulated TNF alpha release in whole bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.10nMAssay Description:Inhibition of P38 alpha MAPKMore data for this Ligand-Target Pair