TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]kianic acid from recombinant GluK1 kainate receptor (unknown origin) expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]kianic acid from recombinant GluK2 kainate receptor (unknown origin) expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 497nMAssay Description:Binding affinity to adrenergic alpha1D receptorMore data for this Ligand-Target Pair
Affinity DataKi: 758nMAssay Description:Binding affinity to adrenergic alpha1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 885nMAssay Description:Binding affinity to adrenergic alpha1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Binding affinity to 5HT1E receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Affinity against adenosine A2 receptor in the brain membranes measured by the displacement of [3H]-CPXMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 3.90E+3nMAssay Description:Affinity against adenosine A2 receptor in the brain membranes measured by the displacement of [3H]-CPXMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+3nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Affinity against adenosine A2 receptor in the brain membranes measured by the displacement of [3H]-CPXMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Homo sapiens (Human))
Hokkaido University
Curated by ChEMBL
Hokkaido University
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity to nicotinic alpha3beta2 receptor receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:Affinity against adenosine A2 receptor in the brain membranes measured by the displacement of [3H]-CPXMore data for this Ligand-Target Pair
Affinity DataKi: 5.60E+3nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.60E+3nMAssay Description:Binding affinity against adenosine A1 receptor of cerebral cortex using [3H]-CPX as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7.30E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 7.60E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 7.70E+3nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Affinity against adenosine A2 receptor in the brain membranes measured by the displacement of [3H]-CPXMore data for this Ligand-Target Pair